IP Library Granted Patent US 6,896,899
Granted Patent B2
US 6,896,899 · App. 10/083,327 · Granted May 24, 2005

Pharmaceutical preparations of glutathione and methods of administration thereof

Assignee: Antioxidant Pharmaceuticals Corp.
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Quick Facts
Patent No.
US 6,896,899
App. No.
10/083,327
Granted
May 24, 2005
Kind
B2
Abstract

A method of increasing glutathione levels in mammalian cells comprising administering an oral bolus of encapsulated pharmaceutically stabilized glutathione in a rapidly dissolving formulation to a mammal on an empty stomach. Pharmaceutical formulations including glutathione are also disclosed.

Claims (25)

1. An pharmaceutical formulation, comprising Glutathione, in combination with an effective amount of one or more of a pharmaceutically acceptable physiologic nitric oxide precursor, and an antimicrobial composition.

2. The formulation according to claim 1 , wherein the formulation acts as a vasodilator through alteration of nitric oxide metabolism.

3. The formulation according to claim 1 , wherein the formulation is effective for treating pathological vasospasm.

4. The formulation according to claim 1 , wherein the formulation is effective for treating sexual dysfunction.

5. The formulation according to claim 1 , in combination with a drug effective to treat congestive heart failure.

6. The formulation according to claim 1 , wherein said formulation is in unit dosage form and comprises in physiologic nitric oxide precursor.

7. The formulation according to claim 6 , wherein the nitric oxide precursor is arginine.

8. The formulation according to claim 6 , wherein said formulation comprises about 500 mg reduced L-glutathione, about 200 mg ascorbic acid, and about 200 mg arginine.

9. The formulation according to claim 1 , wherein the formulation comprises a nitric oxide precursor and an antiviral composition.

10. The formulation according to claim 1 , wherein the nitric oxide precursor comprises an NO 2 functionality.

11. The formulation according to claim 10 , wherein the nitric oxide precursor comprises an organic nitrate.

12. The formulation according to claim 1 , wherein said formulation comprises a pharmacutically acceptable antimicrobial antibiotic agent.

13. The formulation according to claim 1 , wherein said antimicrobial compostion comprises an antimicrobial having activity against mycoplasma infection.

14. The formulation according to claim 1 , wherein said antimicrobial agent comprises an antibiotic in sufficient amount to suppress growth of a microbe and said glutathione is provided in sufficent amount to control free radical reactions associated with the microbe.

15. The pharmaceutical formulation according to claim 1 , wherein said formulation is provided in an oral dosage form.

16. The formulation according to claim 1 , wherein said antimicrobial compostion comprises an aminoglycoside.

17. The formulation according to claim 1 , wherein said antimicrobial compostion comprises a quinolone antibiotic.

18. The formulation according to claim 1 , wherein said formulation is adaptcd to modify vascular tone in an organism administered said formulation.

19. A pharmaccutical composition comprising in combination glutathione, or a pharmaccutically acceptable salt or derivative thereof, and an antiviral or antimicrobial antibiotic agent, said glutathione being present in an effective amount to at least one of: serve as an efffective antioxidant agent; supplement endogenous glutathione consumed as a result of administration of the pharmaccutical composition; alter cardiovascular status of a host; alter a redox status of a bost; and alter a gene expression within a host, and said antimicrobial agent being present in an effective amount to treat or prophylax a microbial-associated condition of the host.

20. The pharmaceutical composition according to claim 19 , comprising, in unit dosage form, glutathione in an amount of at least 250 mg., a sacrificial antioxidant to preserve the glutathione in a reduced state, an effective amount of a pharmaceutically acceptable topoisomerase inhibitor, and a pharmaceutically acceptable physiologic nitric oxide precursor.

21. The pharmaceutical composition according to claim 19 , wherein the antioxidant comprises ascorbic acid.

22. The pharmaceutical composition according to claim 19 , further comprising an antibiotic having activity against mycoplasma infection.

23. The pharmaceutical composition according to claim 19 , wherein said composition is provided in an oral dosage form.

24. The pharmaceutical composition according to claim 19 , comprising an aminoglycoside antibiotic.

25. The pharmaceutical composition according to claim 19 , comprising a quinolone antibiotic.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 14, 2017
From: DEMOPOULOS, HARRY B.; SELIGMAN, MYRON L.
To: ANTIOXIDANT PHARMACEUTICALS CORPORATION
Reel/Frame 041249/0906 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 14, 2017
From: ANTIOXIDANT PHARMACEUTICALS CORPORATION
To: MOLECULAR DEFENSES HOLDINGS, LLC
Reel/Frame 041709/0271 →
Continuity (3)
Continuation 0933194700
Provisional Application 6003410100 · Dec 31, 1996
Related Publication 20020136763A1 · Sep 26, 2002