IP Library Granted Patent US 7,632,499
Granted Patent B2
US 7,632,499 · App. 12/066,838 · Granted Dec 15, 2009

Anti-myostatin antibodies

Assignee: Eli Lilly and Company
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Quick Facts
Patent No.
US 7,632,499
App. No.
12/066,838
Granted
Dec 15, 2009
Kind
B2
Abstract

Anti-myostatin antibodies are identified that are characterized as having high affinity and may be chimeric, humanized or fully human antibodies, immunoconjugates of the antibodies or antigen-binding fragments thereof. The antibodies of the invention are useful for increasing muscle mass, increasing bone density, or for the treatment of various disorders in mammalian and avian species.

Claims (24)

1. An anti-myostatin monoclonal antibody comprising a heavy chain variable region (HCVR) and a light chain variable region (LCVR), wherein said HCVR comprises:

a) a peptide at CDRH1 with SEQ ID NO: 42,

b) a peptide at CDRH2 with SEQ ID NO: 71, and

c) a peptide at CDRH3 with SEQ ID NO: 72,

and wherein said LCVR comprises:

a) a peptide at CDRL1 with SEQ ID NO: 12,

b) a peptide at CDRL2 with SEQ ID NO: 154, and

c) a peptide at CDRL3 with SEQ ID NO: 37.

2. The antibody of claim 1 , wherein the antibody is a full-length antibody, a substantially intact antibody, a Fab fragment, a F(ab′) 2 fragment or a single chain Fv fragment.

3. The anti-myostatin monoclonal antibody of claim 1 , wherein the HCVR comprises:

a) a peptide at CDRH1 with SEQ ID NO: 40,

b) a peptide at CDRH2 with SEQ ID NO: 60, and

c) a peptide at CDRH3 with SEQ ID NO: 72,

and wherein said LCVR comprises:

a) a peptide at CDRL1 with SEQ ID NO: 9,

b) a peptide at CDRL2 with SEQ ID NO: 18, and

c) a peptide at CDRL3 with SEQ ID NO: 34.

4. The antibody of claim 3 , wherein the antibody is a full-length antibody, a substantially intact antibody, a Fab fragment, a F(ab′) 2 fragment or a single chain Fv fragment.

5. An anti-myostatin monoclonal antibody, wherein the LCVR comprises a polypeptide with SEQ ID NO: 98 and the HCVR comprises a polypeptide with SEQ ID NO: 138.

6. The antibody of claim 5 , wherein the antibody is a full-length antibody, a substantially intact antibody, a Fab fragment, a F(ab′) 2 fragment or a single chain Fv fragment.

7. The anti-myostatin monoclonal antibody of claim 5 , wherein the light chain further comprises a constant region polypeptide with SEQ ID NO: 155, and the heavy chain further comprises a constant region polypeptide with SEQ ID NO: 157.

8. A pharmaceutical composition comprising an antibody of claim 1 .

9. A pharmaceutical composition comprising an antibody of claim 3 .

10. A pharmaceutical composition comprising an antibody of claim 5 .

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 2, 2008
From: JONES, BRYAN E.; MITCHELL, PAMELA J.; SMITH, ROSAMUND C.; TOBIAS, LINDA O.; WANG, RONG; KORYTKO, ANDREW I.; DAVIES, JULIAN
To: ELI LILLY AND COMPANY
Reel/Frame 020743/0336 →
Continuity (2)
Provisional Application 6072573800 · Oct 12, 2005
Related Publication 20090131638A1 · May 21, 2009