IP Library Granted Patent US 7,776,895
Granted Patent B2
US 7,776,895 · App. 12/211,322 · Granted Aug 17, 2010

Inhalation devices for delivering phenethanolamine derivatives for the treatment of respiratory diseases

Assignee: Glaxo Group Limited
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 7,776,895
App. No.
12/211,322
Granted
Aug 17, 2010
Kind
B2
Abstract

The invention provides inhalation devices comprising a compound which is 4-{(1R)-2-[(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl)amino]-1-hydroxyethyl}-2-(hydroxymethyl)phenol; or a salt or solvate thereof, inhalation devices comprising formulations and combinations of the compound or a salt or solvate thereof, and methods for the treatment or prophylaxis of a clinical condition in a mammal by employing the inhalation devices.

Claims (9)

1. An inhaler for delivering a pharmaceutically active compound to the lung, said inhaler comprising one or more containers having a dry powder formulation present therein, said dry powder formulation comprising a compound which is 4-{(1R)-2-[(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl)amino]-1-hydroxyethyl}-2-(hydroxymethyl) phenol; or a pharmaceutically acceptable salt thereof.

2. An inhaler according to claim 1 , wherein the compound is present as a pharmaceutically acceptable salt which is a α-phenyl cinnamate salt.

3. An inhaler according to claim 1 , wherein the compound is present as a pharmaceutically acceptable salt which is a 1-naphthoate salt.

4. An inhaler according to claim 1 , wherein the compound is present as a pharmaceutically acceptable salt which is an (R)-mandelate salt.

5. An inhaler according to claim 1 , wherein the compound is present in particles ranging in size from 1 μm to 10 μm.

6. An inhaler according to claim 1 , wherein the dry powder formulation comprises lactose.

7. An inhaler for delivering a pharmaceutically active compound to the lung, said inhaler comprising one or more containers having a dry powder formulation present therein, said dry powder formulation comprising a compound which is 4-{(1R)-2-[(6-{2-[(2,6-dichlorobenzyl) oxy]ethoxy}hexyl)amino]-1-hydroxyethyl}-2-(hydroxymethyl)phenol-triphenyl acetate.

8. An inhaler according to claim 7 , wherein the compound is present in particles ranging in size from 1 μm to 10 μm.

9. An inhaler according to claim 7 , wherein the dry powder formulation comprises lactose.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 1, 2013
From: BOX, PHILIP CHARLES; COE, DIANE MARY; LOOKER, BRIAN EDGAR; MANN, INDERJIT SINGH; PROCOPIOU, PANAYIOTIS ALEXANDROU
To: GLAXO GROUP LIMITED
Reel/Frame 029903/0936 →
Priority Claims (2)
GB 0122201.7 · Sep 14, 2001 · national
GB 0126997.6 · Nov 9, 2001 · national
Continuity (3)
Continuation 1156634600 · Dec 4, 2006
Continuation 1048956900
Related Publication 20090068273A1 · Mar 12, 2009