Granted Patent
B2
US 7,960,399 · App. 11/569,802 · Granted Jun 14, 2011
Quinazolinone derivatives useful as vanilloid antagonists
Assignee:
Novartis AG
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Abstract
The present invention relates to the use of a quinazolinone compound of the formula (I) wherein R 1 , R 2 , R 3 , R 4 , R 5 and m are as defined in the specification and in the claims, in free form or in salt form, and, where possible, in acid addition salt form, as a vanilloid.
Claims (5)
1. A compound of the formula:
in free form or in pharmaceutically acceptable salt form.
2. The compound of claim 1 , wherein the compound is in pharmaceutically acceptable salt form.
3. A pharmaceutical composition comprising a compound of claim 1 , in free form or pharmaceutically acceptable salt form, in association with a pharmaceutical carrier or diluent.
4. The compound of claim 1 , wherein the compound is in free form.
Assignments (6)
INTELLECTUAL PROPERTY SECURITY AGREEMENT
Recorded Dec 23, 2025
From: BAUSCH + LOMB IRELAND LIMITED
To: JPMORGAN CHASE BANK, N.A., AS COLLATERAL AGENT
Reel/Frame 074050/0573 →
INTELLECTUAL PROPERTY SECURITY AGREEMENT
Recorded Dec 23, 2025
From: BAUSCH + LOMB IRELAND LIMITED
To: CITIBANK, N.A., AS NOTES COLLATERAL AGENT
Reel/Frame 074050/0682 →
INTELLECTUAL PROPERTY SECURITY AGREEMENT
Recorded Dec 23, 2025
From: BAUSCH + LOMB IRELAND LIMITED
To: CITIBANK, N.A., AS NOTES COLLATERAL AGENT
Reel/Frame 074050/0709 →
ASSIGNMENT OF ASSIGNOR'S INTEREST
Recorded Dec 6, 2023
From: NOVARTIS AG
To: BAUSCH + LOMB IRELAND LIMITED
Reel/Frame 065790/0208 →
CORRECTIVE ASSIGNMENT TO CORRECT THE ASSIGNOR TO ASSIGNEE PREVIOUSLY RECORDED ON REEL 021429 FRAME 0720. ASSIGNOR(S) HEREBY CONFIRMS THE CORRECT ASSIGNOR TO ASSIGNEE.
Recorded May 8, 2009
From: RITCHIE, TIMOTHY JOHN; CULSHAW, ANDREW JAMES; BRAIN, CHRISTOPHER THOMAS; DZIADULEWICZ, EDWARD KAROL; HART, TERANCE WILLIAM
To: NOVARTIS AG
Reel/Frame 022666/0180 →
ASSIGNMENT OF ASSIGNOR'S INTEREST
Recorded Aug 22, 2008
From: NOVARTIS AG
To: RITCHIE, TIMOTHY JOHN; CULSHAW, ANDREW JAMES; BRAIN, CHRISTOPHER THOMAS; DZIADULEWICZ, EDWARD KAROL; HART, TERANCE WILLIAM
Reel/Frame 021429/0720 →
Priority Claims (1)
GB 0412769.2
· Jun 8, 2004
· national
Continuity (1)