IP Library Granted Patent US 8,067,426
Granted Patent B2
US 8,067,426 · App. 12/537,392 · Granted Nov 29, 2011

6-amino-purin-8-one compounds

Assignee: GlaxoSmithKline LLC
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Quick Facts
Patent No.
US 8,067,426
App. No.
12/537,392
Granted
Nov 29, 2011
Kind
B2
Abstract

Compounds of formula (I): wherein R 1 is C 1-6 alkylamino, C 1-6 alkoxy, or C 3-7 cycloalkyloxy; m is an integer having a value of 3 to 6; n is an integer having a value of 0 to 4; and salts thereof are inducers of human interferon. Compounds which induce human interferon may be useful in the treatment of various disorders, for example the treatment of allergic diseases and other inflammatory conditions for example allergic rhinitis and asthma, the treatment of infectious diseases and cancer, and may also be useful as vaccine adjuvants.

Claims (5)

1. 6-amino-2-{[(1S)-1-methylbutyl]oxy}-9-[5-(1-piperidinyl)pentyl]-7,9-dihydro-8H-purin-8-one, or a salt thereof.

2. 6-amino-2-{[(1S)-1-methylbutyl]oxy}-9-[5-(1-piperidinyl)pentyl]-7,9-dihydro-8H-purin-8-one, or a pharmaceutically acceptable salt thereof.

3. 6-amino-2-{[(1S)-1-methylbutyl]oxy}-9-[5-(1-piperidinyl)pentyl]-7,9-dihydro-8H-purin-8-one as the free base.

4. A pharmaceutical composition comprising a compound according to claim 2 and one or more pharmaceutically acceptable diluents or carriers.

5. A pharmaceutical composition comprising a compound according to claim 3 and one or more pharmaceutically acceptable diluents or carriers.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 28, 2013
From: BIGGADIKE, KEITH; COE, DIANE MARY; LEWELL, XIAO QING; MITCHELL, CHARLOTTE JANE; SMITH, STEPHEN ALLAN; TRIVEDI, NAIMISHA
To: SMITHKLINE BEECHAM CORPORATION
Reel/Frame 030104/0001 →
CHANGE OF NAME Recorded Mar 28, 2013
From: SMITHKLINE BEECHAM CORPORATION
To: GLAXOSMITHKLINE LLC
Reel/Frame 030105/0331 →
Continuity (2)
Provisional Application 61087777 · Aug 11, 2008
Related Publication 20100075995A1 · Mar 25, 2010