IP Library Granted Patent US 8,071,786
Granted Patent B2
US 8,071,786 · App. 12/637,600 · Granted Dec 6, 2011

Indole compounds useful as serotonin selective agents

Assignee: Galenea Corp.
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Quick Facts
Patent No.
US 8,071,786
App. No.
12/637,600
Granted
Dec 6, 2011
Kind
B2
Abstract

Novel indole compounds are disclosed. Also disclosed are methods for using the compounds to treat human and animal disease, pharmaceutical compositions of the compounds, and kits including the compounds.

Claims (23)

1. A compound of formula (I):

wherein:

R is —CH 3 , —CH 2 CH 3 , —CH 2 CH 2 CH 3 , —CH 2 CH 2 CH 2 CH 3 , -cyclopropylmethyl, —CH(CH 3 ) 2 , —SO 2 CH 3 , or —SO 2 CH 2 CH 3 .

2. A compound of formula (II):

wherein:

R is —CH 3 , —CH 2 CH 3 , —CH 2 CH 2 CH 3 , —CH 2 CH 2 F, —CH 2 CH 2 CH 2 CH 3 , -cyclopropylmethyl, —CH(CH 3 ) 2 , —SO 2 CH 3 , or —SO 2 CH 2 CH 3 .

3. A compound of the following formula:

4. A compound of the following formula:

5. A compound of the following formula:

6. The compound of claim 1 , wherein the compound is:

7. The compound of claim 1 , wherein the compound is:

8. The compound of claim 1 , wherein the compound is:

9. The compound of claim 1 , wherein the compound is:

10. The compound of claim 1 , wherein the compound is:

11. The compound of claim 1 , wherein the compound is:

12. The compound of claim 2 , wherein the compound is:

13. The compound of claim 2 , wherein the compound is:

14. The compound of claim 2 , wherein the compound is:

15. The compound of claim 2 , wherein the compound is:

16. The compound of claim 2 , wherein the compound is:

17. The compound of claim 2 , wherein the compound is:

18. The compound of claim 2 , wherein the compound is:

19. The compound of claim 2 , wherein the compound is:

Continuity (2)
Continuation 11237318 · Sep 27, 2005
Related Publication 20100137616A1 · Jun 3, 2010