IP Library Granted Patent US 8,143,217
Granted Patent B2
US 8,143,217 · App. 12/067,314 · Granted Mar 27, 2012

Use of DPP-IV inhibitor to reduce hypoglycemic events

Assignee: Novartis AG
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Quick Facts
Patent No.
US 8,143,217
App. No.
12/067,314
Granted
Mar 27, 2012
Kind
B2
Abstract

The invention relates to a method to reduce the hypoglycemic events, especially sever hypoglycemic events resulting from insulin treatment, wherein the patient is treated with a Dipeptidyl peptidase IV inhibitor (DPP-IV inhibitor) or a pharmaceutically acceptable salt thereof.

Claims (12)

1. A method for reducing hypoglycemic events or severe hypoglycemic events in a patient suffering from hyperglycemia, diabetes mellitus, insulin-dependent diabetes mellitus (IDDM), non-insulin-dependent diabetes mellitus (NIDDM), type A insulin resistance, Impaired Glucose Metabolism (IGM), Impaired Fasting Glucose (IFG) or Impaired Glucose Tolerance (IGT), said method comprising:

i) selecting a patient treated by insulin and showing hypoglycemic episodes or severe hypoglycemic events; and

ii) administering vildagliptin or a salt thereof, in combination with insulin to said patient.

2. The method according to claim 1 , wherein the vildagliptin and insulin are administered simultaneously or sequentially, and in any order.

3. The method of claim 1 wherein the vildagliptin is administered in amounts of between 25 and 150 mg per day.

4. The method according to claim 1 wherein the patient is under treatment with an additional one, two or three antidiabetic compounds.

5. The method of claim 4 , wherein the additional antidiabetic compound is selected from metformin, nateglinide, glitazones, sulfonylureas, GLP-1 or GLP-1 analogues, and cannabinoid receptor-1 (CB1) antagonists.

6. The method of claim 4 , wherein the patient is under treatment with an additional two antidiabetic compounds selected from: metformin and a sulfonylurea, metformin and a glitazone, metformin and a GLP-1 analogue, metformin and a CB1 antagonist, a glitazone and a sulfonylurea, and a GLP-1 analogue and a sulfonylurea.

7. The method of claim 1 wherein the hypoglycemic events or severe hypoglycemic events are resulting from insulin treatment or from treatment with insulin and at least one additional antidiabetic compound.

8. The method according to claim 1 wherein between 25 and 200 mg of vildagliptin or a salt thereof, is administered daily.

9. The method of claim 5 , wherein the glitazone is pioglitazone or rosiglitazone.

10. The method of claim 5 , wherein the GLP-1 analogue is exendin-4.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 13, 2011
From: BALKAN, BOERK; HOLMES, DAVID GRENVILLE; HUGHES, THOMAS EDWARD; VILLHAUER, EDWIN BERNARD
To: NOVARTIS AG
Reel/Frame 027372/0203 →
Continuity (3)
Provisional Application 60718856 · Sep 20, 2005
Provisional Application 60786755 · Mar 28, 2006
Related Publication 20080300171A1 · Dec 4, 2008