IP Library Granted Patent US 8,354,515
Granted Patent B2
US 8,354,515 · App. 13/126,320 · Granted Jan 15, 2013

Oligonucleotide derivative, labeling agent and use for labeling agent

Inventors: Yoshihito Ueno (Gifu, JP); Yukio Kitade (Gifu, JP)
Assignee: Japan Science and Technology Agency
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Quick Facts
Patent No.
US 8,354,515
App. No.
13/126,320
Granted
Jan 15, 2013
Kind
B2
Abstract

A labeling agent comprising a plurality of nucleotide derivative units represented by Formula (1) below: (where, Z represents a nitrogen atom or CH, Y represents an uncondensed aromatic hydrocarbon group or condensed polycyclic hydrocarbon group, X 1 represents O, S or Se, and X 2 represents SH (or S − ), Se − , a C 1-4 alkyl or a morpholino group).

Claims (16)

1. A labeling agent comprising a plurality of nucleotide derivative units represented by Formula (1) below:

(where, Z represents a nitrogen atom or CH, Y represents an uncondensed aromatic hydrocarbon group or condensed polycyclic hydrocarbon group other than naturally occurring base having purine structure or pyrimidine structure, X 1 represents O, S or Se, and X 2 represents SH (or S − ), Se − , or a C 1-4 alkyl group or morpholino group).

2. The labeling agent according to claim 1 , wherein said Y is a condensed polycyclic hydrocarbon group.

3. The labeling agent according to claim 2 , wherein said Y is selected from a group consisting of naphthalene, phenathrene, pyrene and perylene.

4. The labeling agent according to claim 1 , comprising a plurality of said nucleotide derivative units in a continuous series.

5. The labeling agent according to claim 1 , comprising a plurality of said nucleotide derivative units, with linker units in between.

6. The labeling agent according to claim 1 , wherein said multiple nucleotide units are two nucleotide derivative units in which said Y is the same or different, and are provided in a continuous series.

7. A set of labeling agents comprising two or more labeling agents each provided with a plurality of nucleotide derivative units represented by Formula (1) below:

(where, Z represents a nitrogen atom or CH, Y represents an uncondensed aromatic hydrocarbon group or condensed polycyclic hydrocarbon group other than naturally occurring base having purine structure or pyrimidine structure, X 1 represents O, S or Se, and X 2 represents SH (or S − ), Se − , or a C 1-4 alkyl group or morpholino group), wherein the sequence of said Y in said plurality of nucleotide derivative units is different for each of the labeling agents.

8. The set of labeling agents according to claim 7 , further comprising a labeling agent provided with one of the nucleotide derivative units represented by Formula (1) above.

9. An oligonucleotide probe comprising a plurality of nucleotide derivative units represented by Formula (1) below:

(where, Z represents a nitrogen atom or CH, Y represents an uncondensed aromatic hydrocarbon group or condensed polycyclic hydrocarbon group other than naturally occurring base having purine structure or pyrimidine structure, X 1 represents O, S or Se, and X 2 represents SH (or S − ), Se − , or a C 1-4 alkyl group or morpholino group).

10. The oligonucleotide probe according to claim 9 , comprising said plurality of nucleotide derivative units at the 3′ terminal end or 5′ terminal end.

11. An oligonucleotide probe set comprising two or more oligonucleotide probes each provided with a plurality of nucleotide derivative units represented by Formula (1) below:

(where, Z represents a nitrogen atom or CH, Y represents an uncondensed aromatic hydrocarbon group or condensed polycyclic hydrocarbon group other than naturally occurring base having purine structure or pyrimidine structure, X 1 represents O, S or Se, and X 2 represents SH (or S − ), Se − or a C 1-4 alkyl group or morpholino group), wherein the sequence of said Y in said plurality of nucleotide derivative units is different for each of the probes.

12. The oligonucleotide probe set according to claim 11 , further comprising a labeling agent provided with one of the nucleotide derivative units represented by Formula (1).

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 23, 2011
From: UENO, YOSHIHITO; KITADE, YUKIO
To: JAPAN SCIENCE AND TECHNOLOGY AGENCY
Reel/Frame 026509/0868 →
Priority Claims (1)
JP 2008-292815 · Nov 14, 2008 · national
Continuity (1)
Related Publication 20120126175A1 · May 24, 2012