IP Library Granted Patent US 8,383,823
Granted Patent B2
US 8,383,823 · App. 12/143,484 · Granted Feb 26, 2013

Substituted N-aryl pyridinones

Inventors: Thomas G. Gant (Carlsbad, CA); Sepehr Sarshar (Cardiff by the Sea, CA)
Assignee: Auspex Pharmaceuticals
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Quick Facts
Patent No.
US 8,383,823
App. No.
12/143,484
Granted
Feb 26, 2013
Kind
B2
Abstract

Disclosed herein are substituted N-Aryl pyridinone fibrotic inhibitors and/or collagen infiltration modulators of Formula I, process of preparation thereof, pharmaceutical compositions thereof, and methods of use thereof.

Claims (10)

1. A compound having the structural formula:

or a pharmaceutically acceptable salt thereof.

2. The compound as recited in claim 1 , wherein each of said positions represented as D has deuterium enrichment of at least 98%.

3. The compound as recited in claim 1 , wherein each of said positions represented as D has deuterium enrichment of at least 90%.

4. The compound as recited in claim 1 , wherein each of said positions represented as D has deuterium enrichment of at least 50%.

5. The compound as recited in claim 1 , wherein each of said positions represented as D has deuterium enrichment of at least 20%.

6. The compound as recited in claim 1 , wherein each of said positions represented as D has deuterium enrichment of at least 10%.

7. The compound as recited in claim 1 , wherein each of said positions represented as D has deuterium enrichment of at least 5%.

8. The compound as recited in claim 1 , wherein each of said positions represented as D has deuterium enrichment of at least 1%.

9. A pharmaceutical composition comprising the compound as recited in claim 1 and one or more pharmaceutically acceptable carriers.

Assignments (4)
CORRECTIVE ASSIGNMENT TO CORRECT THE ASSIGNEE NAME PREVIOUSLY RECORDED ON REEL 050487 FRAME 0946. ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNMENT.. Recorded Nov 1, 2019
From: PURETECH HEALTH LLC
To: PURETECH LYT 100, INC.
Reel/Frame 050902/0278 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 25, 2019
From: PURETECH HEALTH LLC
To: PURETECH LYT-100, INC.
Reel/Frame 050487/0946 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 23, 2019
From: AUSPEX PHARMACEUTICALS, INC.
To: PURETECH HEALTH LLC
Reel/Frame 050147/0568 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 18, 2008
From: GANT, THOMAS G.; SARSHAR, SEPEHR
To: AUSPEX PHARMACEUTICALS, INC.
Reel/Frame 021260/0797 →
Continuity (2)
Provisional Application 60945136 · Jun 20, 2007
Related Publication 20080319026A1 · Dec 25, 2008