IP Library Granted Patent US 8,410,145
Granted Patent B2
US 8,410,145 · App. 12/808,847 · Granted Apr 2, 2013

Insecticidal compounds

Inventors: Pierre Joseph Marcel Jung (Stein, CH); Peter Renold (Stein, CH)
Assignee: Syngenta Crop Protection LLC
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Quick Facts
Patent No.
US 8,410,145
App. No.
12/808,847
Granted
Apr 2, 2013
Kind
B2
Abstract

A compound of formula (I): wherein A 1 , A 2 , A 3 , A 4 , G 1 , R 1 , R 2 , R 3 and R 4 are as defined in claim 1 ; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of Formula (I), to insecticidal, acaricidal, molluscicidal or nematicidal compositions comprising them and to methods of using them to combat and control insect, acarine, mollusc or nematode pests.

Claims (33)

1. A compound of formula (I)

wherein

A 1 , A 2 , and A 3 are independently of one another C—H, C—R 5 , or nitrogen, provided that no more than two of A 1 , A 2 , and A 3 are nitrogen;

A 4 is C—CN;

G 1 is oxygen or sulfur;

R 1 is C 1 -C 6 alkyl, C 1 -C 6 haloalkyl, C 1 -C 3 alkoxy-C 1 -C 3 alkyl-, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, C 1 -C 6 alkoxycarbonyl-, aryl-C 1 -C 6 alkyl- or aryl-C 1 -C 6 alkyl- substituted by one to three R 6 , heterocyclyl-C 1 -C 6 alkyl- or heterocyclyl-C 1 -C 6 alkyl- substituted by one to three R 6 ; or

R 1 is aryl or aryl substituted by one to three R 6 , or

R 1 is heterocyclyl or heterocyclyl substituted by one to three R 6 ;

R 2 is hydrogen, C 1 -C 6 alkyl, C 1 -C 6 alkylcarbonyl-, or C 1 -C 6 alkoxycarbonyl-;

R 3 is C 1 -C 6 haloalkyl;

R 4 is aryl or aryl substituted by one to three R 7 , or heterocyclyl or heterocyclyl substituted by one to three R 7 ;

each R 5 is independently halogen, cyano, nitro, C 1 -C 6 alkyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, or C 1 -C 6 alkoxycarbonyl-;

each R 6 is independently halogen, cyano, nitro, C 1 -C 6 alkyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, C 1 -C 6 alkylthio-, C 1 -C 6 haloalkylthio-, C 1 -C 6 alkylsulfinyl-, C 1 -C 6 haloalkylsulfinyl-, C 1 -C 6 alkylsulfonyl-, C 1 -C 6 haloalkylsulfonyl-, or C 1 -C 6 alkoxycarbonyl-; and

each R 7 is independently halogen, cyano, nitro, C 1 -C 6 alkyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, or C 1 -C 6 alkoxycarbonyl-; or a salt or N-oxide thereof.

2. A compound according to claim 1 wherein A 1 is C—H or C—R 5 .

3. A compound according to claim 1 wherein A 2 is C—H or C—R 5 .

4. A compound according to claim 1 wherein A 3 is C—H or C—R 5 .

5. A compound according to claim 1 wherein G 1 is oxygen.

6. A compound according to claim 1 wherein R 1 is C 1 -C 6 alkyl, C 1 -C 6 haloalkyl, C 1 -C 3 alkoxy-C 1 -C 3 alkyl-, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, aryl-C 1 -C 6 alkyl- or aryl-C 1 -C 6 alkyl- substituted by one to three R 6 , aryl or aryl substituted by one to three R 6 , or heterocyclyl or heterocyclyl substituted by one to three R 6 .

7. A compound according to claim 1 wherein R 2 is hydrogen, methyl, ethyl, methylcarbonyl-, or methoxycarbonyl-.

8. A compound according to claim 1 wherein R 3 is chlorodifluoromethyl or trifluoromethyl.

9. A compound according to claim 1 wherein R 4 is aryl or aryl substituted by one to three R 7 .

10. A compound according to claim 1 wherein each R 5 is independently bromo, chloro, fluoro, cyano, nitro, methyl, ethyl, trifluoromethyl, methoxy, difluoromethoxy, trifluoromethoxy, or methoxycarbonyl.

11. A method of combating and controlling insects, acarines, molluscs or nematodes which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, molluscicidally or nematicidally effective amount of a compound of formula (I) as defined in claim 1 .

12. An insecticidal, acaricidal, molluscicidal or nematicidal composition comprising an insecticidally, acaricidally, molluscicidally or nematicidally effective amount of a compound of formula (I) as defined in claim 1 .

13. An insecticidal, acaricidal, molluscicidal or nematicidal composition according to claim 12 , wherein the composition contains one or more additional active ingredients.

14. A compound according to claim 1 wherein:

A 1 , A 2 , and A 3 are each C—H;

G 1 is oxygen; and

R 1 is aryl or aryl substituted by one to three R 6 .

15. A compound according to claim 14 wherein R 2 is hydrogen.

16. An insecticidal, acaricidal, molluscicidal or nematicidal composition comprising an insecticidally, acaricidally, molluscicidally or nematicidally effective amount of a compound of formula (I) as defined in claim 14 .

17. An insecticidal, acaricidal, molluscicidal or nematicidal composition comprising an insecticidally, acaricidally, molluscicidally or nematicidally effective amount of a compound of formula (I) as defined in claim 15 .

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 19, 2012
From: JUNG, PIERRE JOSEPH MARCEL; RENOLD, PETER
To: SYNGENTA CROP PROTECTION LLC
Reel/Frame 028403/0011 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 12, 2012
From: JUNG, PIERRE JOSEPH MARCEL; RENOLD, PETER
To: SYNGENTA CROP PROTECTION LLC
Reel/Frame 028358/0021 →
Priority Claims (2)
GB 0724757.0 · Dec 19, 2007 · national
GB 0808471.7 · May 9, 2008 · national
Continuity (1)
Related Publication 20100273832A1 · Oct 28, 2010