IP Library Granted Patent US 8,415,355
Granted Patent B2
US 8,415,355 · App. 12/545,322 · Granted Apr 9, 2013

Pyrrolopyrimidine compounds and their uses

Inventors: Christopher Thomas Brain (Cambridge, MA); Moo Je Sung (Cambridge, MA); Bharat Lagu (Acton, MA)
Assignees: Novartis AG; Astex Therapeutics Ltd.
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Quick Facts
Patent No.
US 8,415,355
App. No.
12/545,322
Granted
Apr 9, 2013
Kind
B2
Abstract

The present invention relates to compounds of formula (I) and to pharmaceutically acceptable salts and pharmaceutical compositions thereof. The present invention also relates to use of the compounds of formula (I) in modulating the activity of protein kinases and in the treatment of disease, particularly a disease, disorder or syndrome associated with CDK 4 inhibition.

Claims (7)

1. A compound 7-Cyclopentyl-2-(5-piperazin-1-yl-pyridin-2-ylamino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide of the formula

or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising a compound according to claim 1 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier.

3. The composition according to claim 2 suitable for oral administration.

4. A compound 7-Cyclopentyl-2-(5-piperazin-1-yl-pyridin-2-ylamino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide of the formula

5. A pharmaceutical composition comprising a compound according to claim 4 and a pharmaceutically acceptable carrier.

6. The composition according to claim 5 suitable for oral administration.

Assignments (6)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 15, 2021
From: NOVARTIS AG
To: NOVARTIS PHARMACEUTICALS CORPORATION
Reel/Frame 056549/0645 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 6, 2013
From: ASTEX THERAPEUTICS LIMITED; NOVARTIS AG
To: NOVARTIS AG; ASTEX THERAPEUTICS LIMITED
Reel/Frame 029934/0265 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 22, 2012
From: LAGU, BHARAT
To: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC.
Reel/Frame 029164/0608 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 22, 2012
From: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC.
To: NOVARTIS AG
Reel/Frame 029164/0683 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 20, 2011
From: BESONG, GILBERT; CONGREVE, MILES STUART; DAGOSTIN, CLAUDIO; HOWARD, STEVEN; MORTENSON, PAUL; WOODHEAD, STEVEN
To: ASTEX THERAPEUTICS LTD.
Reel/Frame 026621/0725 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 20, 2011
From: BRAIN, CHRISTOPHER THOMAS; BROOKS, CLINTON A.; HE, GUO; HOU, YING; LI, YUE; LU, YIPIN; SMITH, TROY; SUNG, MOO JE; WRONA, WOJCIECH
To: NOVARTIS AG
Reel/Frame 026621/0909 →
Continuity (2)
Provisional Application 61091037 · Aug 22, 2008
Related Publication 20100105653A1 · Apr 29, 2010