IP Library Granted Patent US 8,415,387
Granted Patent B2
US 8,415,387 · App. 12/619,412 · Granted Apr 9, 2013

Modulators of ATP-binding cassette transporters

Inventors: Sara S. Hadida Ruah (La Jolla, CA); Peter D. J. Grootenhuis (San Diego, CA); Mark T Miller (San Diego, CA); Jason McCartney (Cardiff By The Sea, CA); Fredrick van Goor (San Diego, CA); Mehdi Michel Djamel Numa (San Diego, CA); Jinglan Zhou (San Diego, CA); Brian Bear (Oceanside, CA)
Assignee: Vertex Pharmaceuticals Incorporated
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 8,415,387
App. No.
12/619,412
Granted
Apr 9, 2013
Kind
B2
Abstract

Compounds of the present invention and pharmaceutically acceptable compositions thereof, are useful as modulators of ATP-Binding Cassette (“ABC”) transporters or fragments thereof, including Cystic Fibrosis Transmembrane Conductance Regulator (“CFTR”). The present invention also relates to methods of treating ABC transporter mediated diseases using compounds of the present invention.

Claims (4)

1. A method of treating a condition, disease, or disorder in a patient implicated by CFTR activity, wherein said condition, disease, or disorder is selected from cystic fibrosis, hereditary emphysema, chronic obstructive pulmonary disease (COPD) and dry eye disease, comprising the step of administering to said patient a compound having the formula:

or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 , wherein said condition, disease, or disorder is cystic fibrosis, hereditary emphysema, or COPD.

3. The method of claim 1 , wherein said condition, disease, or disorder is cystic fibrosis.

Assignments (5)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 21, 2018
From: HADIDA RUAH, SARA S.; GROOTENHUIS, PETER D.J.; VAN GOOR, FREDRICK; ZHOU, JINGLAN; BEAR, BRIAN; MILLER, MARK T.; MCCARTNEY, JASON; NUMA, MEHDI MICHEL DJAMEL
To: VERTEX PHARMACEUTICALS INCORPORATED
Reel/Frame 045305/0447 →
RELEASE OF SECURITY INTEREST Recorded Oct 14, 2016
From: MACQUARIE US TRADING LLC
To: VERTEX PHARMACEUTICALS INCORPORATED; VERTEX PHARMACEUTICALS (SAN DIEGO) LLC
Reel/Frame 040357/0001 →
ASSIGNEE CHANGE OF ADDRESS Recorded Feb 11, 2016
From: VERTEX PHARMACEUTICALS INCORPORATED
To: VERTEX PHARMACEUTICALS INCORPORATED
Reel/Frame 037781/0332 →
SECURITY INTEREST Recorded Jul 10, 2014
From: VERTEX PHARMACEUTICALS INCORPORATED; VERTEX PHARMACEUTICALS (SAN DIEGO) LLC
To: MACQUARIE US TRADING LLC
Reel/Frame 033292/0311 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 4, 2012
From: HADIDA RUAH, SARA S.; GROOTENHUIS, PETER D.J.; VAN GOOR, FREDRICK; ZHOU, JINGLAN; BEAR, BRIAN; MILLER, MARK T.; MCCARTNEY, JASON; NUMA, MEHDI MICHEL JAMEL
To: VERTEX PHARMACEUTICALS INCORPORATED
Reel/Frame 028157/0361 →
Continuity (4)
Division 10975297 · Oct 18, 2007
Continuation In Part 11786001 · Apr 9, 2007
Provisional Application 60790459 · Apr 7, 2006
Related Publication 20100113555A1 · May 6, 2010