IP Library Granted Patent US 9,522,127
Granted Patent B2
US 9,522,127 · App. 14/047,391 · Granted Dec 20, 2016

Use of histone deacetylase inhibitors for the care of philadelphia-negative myeloproliferative syndromes

Inventors: Tiziano Oldoni (Rho, IT); Paolo Mascagni (Villasanta, IT); Alessandro Rambaldi (Bergamo, IT); Tiziano Barbui (Bergamo, IT)
Assignee: ITALFARMACO SPA
A61K31/167A61K31/00A61K31/16A61K31/18A61K45/06
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Quick Facts
Patent No.
US 9,522,127
App. No.
14/047,391
Granted
Dec 20, 2016
Kind
B2
Abstract

Method of treating Philadelphia-negative myeloproliferative syndromes in a patient suffering from such syndromes. The method is carried out by administering to the patient diethyl-[6-(4-hydroxycarbamoyl-phenylcarbamoyloxymethyl)-naphthalen-2-yl -methyl]-ammonium chloride, or other pharmaceutically acceptable salts and/or solvates, in a daily dosage amount of from 10 to 150 mg per patient.

Claims (9)

1. Method of treating Philadelphia-negative myeloproliferative syndromes in a patient suffering from said syndromes, said method comprising administering to said patient diethyl-[6-(4-hydroxycarbamoyl-phenylcarbamoyloxymethyl)-naphthalen-2-yl-methyl]-ammonium chloride, or other pharmaceutically acceptable salts and/or solvates, and at least one other cytostatic active principle, wherein said diethyl-[6-(4-hydroxycarbamoyl-phenylcarbamoyloxymethyl)-naphthalen-2-yl-methyl]-ammonium chloride, or other pharmaceutically acceptable salts and/or solvates thereof is administered in a daily dosage amount of from 50 to 150 mg per patient.

2. Method according to claim 1 , wherein said diethyl-[6-(4-hydroxycarbamoyl-phenylcarbamoyloxymethyl)-naphthalen-2-yl-methyl]-ammonium chloride is in monohydrate form.

3. Method according to claim 1 , wherein said diethyl[6-(4-hydroxycarbamoyl-phenylcarbamoyloxymethyl)-naphthalen-2-yl-methyl]-ammonium chloride is in monohydrate crystal form.

4. Method according to claim 1 , wherein said Philadelphia-negative myeloproliferative syndrome is polycythemia vera.

5. Method according to claim 1 , wherein said Philadelphia-negative myeloproliferative syndrome is essential thrombocythemia.

6. Method according to claim 1 , wherein said Philadelphia-negative myeloproliferative syndrome is primary myeofibrosis.

7. Method according to claim 1 , wherein said Philadelphia-negative myeloproliferative syndrome is secondary myelofibrosis.

8. Method according to claim 1 , wherein said at least one other cytostatic active principle is selected from the group consisting of hydroxyurea and pipobroman.

9. Method according to claim 1 , wherein said daily dosage is from 50 to 100 mg per patient.

Continuity (4)
Division 13064450 · Mar 25, 2011
Continuation PCTEP2009062214 · Sep 21, 2009
Provisional Application 61193283 · Nov 13, 2008
Related Publication 20140039059A1 · Feb 6, 2014