Fused heterocyclic compound and pest control application thereof
Provided are: a fused heterocyclic compound by formula (1) or an N-oxide thereof, having excellent control effects against pests: a pest control composition containing the abovementioned compound and an inert carrier; and a pest control method for applying an effective dose of the abovementioned compound to a pest or pest habitat.
1. A fused heterocyclic compound represented by formula (1);
wherein
R 1 represents a hydrogen atom, a C1-C3 alkyl group which may be optionally substituted with one or more halogen atom(s), a halogen atom, a C1-C3 alkoxy group, a C2-C4 alkoxycarbonyl group, a S(O) m R 2 , a NR 3 R 4 , a nitro group or a cyano group;
R 2 represents a C1-C3 alkyl group;
R 3 and R 4 are the same or different from each other, and each represents a hydrogen atom or a C1-C3 alkyl group;
n is 0, 1 or 2; and
m is 0, 1 or 2
or N-oxide thereof.
2. The compound according to claim 1 wherein R 1 represents a hydrogen atom, a C1-C3 alkyl group which may be optionally substituted with one or more halogen atom(s), a halogen atom, a C1-C3 alkoxy group, or a S(O) m R 2 .
3. The compound according to claim 1 wherein R 1 represents a hydrogen atom, a halogen atom, a C1-C3 perfluoroalkyl group, a C1-C3 alkoxy group, or a S(O) 1 R 2 .
4. The compound according to claim 1 wherein R 1 represents a hydrogen atom, a chlorine atom, a bromine atom, a methyl group, a trifluoromethyl group, a methoxy group, a methylsulfanyl group, a methylsulfinyl group or a methylsulfonyl group.
5. The compound according to claim 1 wherein R 1 represents a hydrogen atom, a chlorine atom, a bromine atom, a trifluoromethyl group, a methoxy group, a methylsulfanyl group or a methylsulfonyl group.
6. The compound according to claim 1 wherein R 1 represents a hydrogen atom.
7. The compound according to claim 1 , wherein n is 2.
8. A composition for controlling a pest comprising the compound according to claim 1 and an inert carrier.
9. A method for controlling a pest, which comprises a step of applying an effective amount of the compound according claim 1 to a pest or a habitat where the pest lives.
10. A method for producing a fused heterocyclic compound represented by formula (1),
comprising a step of reacting a compound represented by formula (M1) with a compound represented by formula (M2):
wherein
R 1 represents a hydrogen atom, a C1-C3 alkyl group which may be optionally substituted with one or more halogen atom(s), a halogen atom, a C1-C3 alkoxy group, a C2-C4 alkoxycarbonyl group, a S(O) m R 2 , a NR 3 R 4 , a nitro group or a cyano group;
R 2 represents a C1-C3 alkyl group;
R 3 and R 4 are the same or different from each other, and each represents a hydrogen atom or a C1-C3 alkyl group;
n is 0, 1 or 2;
m is 0, 1 or 2; and
X is a halogen atom.
11. The method according to claim 10 wherein the step of reacting the compound represented by formula (M1) with the compound represented by formula (M2) is carried out in presence of base.
12. The method according to claim 11 wherein the base is alkali metal hydride, alkaline-earth metal hydride, or alkali metal carbonate.