IP Library Granted Patent US 9,670,205
Granted Patent B2
US 9,670,205 · App. 15/059,070 · Granted Jun 6, 2017

Toll like receptor modulator compounds

Inventors: Evangelos Aktoudianakis (Redwood City, CA); Gregory Chin (San Francisco, CA); Richard L. Mackman (Millbrae, CA); Samuel E. Metobo (Newark, CA); Michael R. Mish (Foster City, CA); Hyung-jung Pyun (Fremont, CA); Jeff Zablocki (Los Altos, CA)
Assignee: GILEAD SCIENCES, INC.
C07D471/04
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Quick Facts
Patent No.
US 9,670,205
App. No.
15/059,070
Granted
Jun 6, 2017
Kind
B2
Abstract

The present disclosure relates generally to toll like receptor modulator compounds, such as diamino pyrido[3,2 D]pyrimidine compounds and pharmaceutical compositions which, among other things, modulate toll-like receptors (e.g. TLR-8), and methods of making and using them.

Claims (20)

1. A compound which is

or a pharmaceutically acceptable salt thereof.

2. A compound which is

3. A pharmaceutical composition comprising the compound of claim 1 or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

4. A pharmaceutical composition comprising the compound of claim 2 , and a pharmaceutically acceptable excipient.

5. A compound which is

or a pharmaceutically acceptable salt thereof.

6. A compound which is

7. A pharmaceutical composition comprising the compound of claim 5 or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

8. A pharmaceutical composition comprising the compound of claim 6 , and a pharmaceutically acceptable excipient.

9. A compound which is

or a pharmaceutically acceptable salt thereof.

10. A compound which is

11. A pharmaceutical composition comprising the compound of claim 9 or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

12. A pharmaceutical composition comprising the compound of claim 10 , and a pharmaceutically acceptable excipient.

13. A compound which is

or a pharmaceutically acceptable salt thereof.

14. A compound which is

15. A pharmaceutical composition comprising the compound of claim 13 or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

16. A pharmaceutical composition comprising the compound of claim 14 , and a pharmaceutically acceptable excipient.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 4, 2016
From: AKTOUDIANAKIS, EVANGELOS; CHIN, GREGORY; MACKMAN, RICHARD L.; METOBO, SAMUEL E.; MISH, MICHAEL R.; PYUN, HYUNG-JUNG; ZABLOCKI, JEFF
To: GILEAD SCIENCES, INC.
Reel/Frame 037898/0322 →
Continuity (3)
Provisional Application 62250403 · Nov 3, 2015
Provisional Application 62128397 · Mar 4, 2015
Related Publication 20160289229A1 · Oct 6, 2016