IP Library Granted Patent US 9,844,561
Granted Patent B2
US 9,844,561 · App. 14/855,293 · Granted Dec 19, 2017

Administration of nicotinamide mononucleotide in the treatment of disease

Inventors: Shin-ichiro Imai (Saint Louis, MO); Rajendra Apte (Clayton, MO)
Assignee: Washington University
A61K31/706A61K9/0014A61K9/0048A61K9/0053A61K31/455A61K31/7064
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Quick Facts
Patent No.
US 9,844,561
App. No.
14/855,293
Granted
Dec 19, 2017
Kind
B2
Abstract

Disclosed are methods and compositions related to methods of treating, ameliorating, mitigating, slowing, arresting, preventing or reversing various diseases and conditions, including age-related obesity, age-related increases in blood lipid levels, age-related decreases in insulin sensitivity, age-related decreases in memory function, and age-related changes in eye function such as macular degeneration. The methods comprise administering nicotinamide mononucleotide (NMN) to a subject. In some embodiments, the administration can be oral administration. Also disclosed are pharmaceutical compositions comprising NMN.

Claims (18)

1. A method of treating photoreceptor degeneration in a subject, comprising: administering to a subject in need of treatment a pharmaceutically effective amount of nicotinamide mononucleotide (NMN) or a salt or prodrug thereof.

2. A method in accordance with claim 1 , wherein the NMN or salt or prodrug thereof is administered orally in a pharmaceutically acceptable formulation selected from the group consisting of a pill, a tablet, a caplet, a capsule, a chewable tablet, a quick dissolve tablet, a powder, a granule, an effervescent tablet, a hard gelatin capsule, a soft gelatin capsule, a non-aqueous liquid, an aqueous liquid, a suspension, a solution, an emulsion, a syrup, a sterilized aqueous suspension, a sterilized aqueous solution, a non-aqueous suspension, a non-aqueous solution, and a lyophilized formulation.

3. A method in accordance with claim 1 , wherein the administering comprises intraocular injection.

4. A method in accordance with claim 1 , wherein the administering comprises topical administration to the eye.

5. A method in accordance with claim 1 , wherein the administering comprises administering the NMN, salt or prodrug thereof in a controlled release formulation.

6. A method in accordance with claim 1 , wherein the photoreceptor degeneration comprises a decline in or loss of photoreceptor function.

7. A method in accordance with claim 6 , wherein the photoreceptor degeneration is selected from the group consisting of retinitis pigmentosa (RP), Leber's congenital amaurosis (LCA), rod dystrophy, cone dystrophy, rod-cone dystrophy, cone-rod dystrophy, age-related macular degeneration and photoreceptor degeneration following retinal detachment.

8. A method in accordance with claim 1 , wherein the photoreceptor degeneration comprises photoreceptor degeneration resulting from a reduction in NAD biosynthesis.

9. A method in accordance with claim 1 , wherein the photoreceptor degeneration is associated with a retinal injury.

10. A method in accordance with claim 1 , wherein the photoreceptor degeneration comprises mitochondrial dysfunction.

11. A method in accordance with claim 1 , wherein the subject is a mammal.

12. A method in accordance with claim 1 , wherein the subject is a human.

13. A method of improving photoreceptor cell function in a mammalian subject, comprising administering to a subject in need of treatment a pharmaceutically effective amount of nicotinamide mononucleotide (NMN) or a salt or prodrug thereof.

14. A method in accordance with claim 13 , wherein the NMN or salt or prodrug thereof is administered orally in a pharmaceutically acceptable formulation selected from the group consisting of a pill, a tablet, a caplet, a capsule, a chewable tablet, a quick dissolve tablet, a powder, a granule, an effervescent tablet, a hard gelatin capsule, a soft gelatin capsule, a non-aqueous liquid, an aqueous liquid, a suspension, a solution, an emulsion, a syrup, a sterilized aqueous suspension, a sterilized aqueous solution, a non-aqueous suspension, a non-aqueous solution, and a lyophilized formulation.

15. A method of ameliorating age-associated decline in photoreceptor cell function in a subject, comprising administering to a subject in need of treatment a pharmaceutically effective amount of nicotinamide mononucleotide (NMN) or a salt or prodrug thereof.

16. A method in accordance with claim 15 , wherein the NMN or salt or prodrug thereof is administered orally in a pharmaceutically acceptable formulation selected from the group consisting of a pill, a tablet, a caplet, a capsule, a chewable tablet, a quick dissolve tablet, a powder, a granule, an effervescent tablet, a hard gelatin capsule, a soft gelatin capsule, a non-aqueous liquid, an aqueous liquid, a suspension, a solution, an emulsion, a syrup, a sterilized aqueous suspension, a sterilized aqueous solution, a non-aqueous suspension, a non-aqueous solution, and a lyophilized formulation.

17. A method in accordance with claim 13 , wherein the improving photoreceptor cell function comprises improving rod cell function.

18. A method in accordance with claim 13 , wherein the improving photoreceptor cell function comprises improving cone cell function.

Assignments (2)
CONFIRMATORY LICENSE Recorded Nov 3, 2022
From: WASHINGTON UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 061878/0761 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 22, 2015
From: IMAI, SHIN-ICHIRO; APTE, RAJENDRA
To: WASHINGTON UNIVERSITY
Reel/Frame 036619/0572 →
Continuity (4)
Continuation PCTUS2014030920 · Mar 17, 2014
Provisional Application 61801188 · Mar 15, 2013
Provisional Application 61947387 · Mar 3, 2014
Related Publication 20160022712A1 · Jan 28, 2016