IP Library Granted Patent US 9,932,302
Granted Patent B1
US 9,932,302 · App. 14/519,679 · Granted Apr 3, 2018

N-phenyl and N-benzyl enaminones and methods for using same

Inventors: Patrice L. Jackson-Ayotunde (Salisbury, MD); Tawes Harper (East New Market, MD)
Assignee: University of Maryland Eastern Shore
C07C311/29A61J1/05C07C233/76C07C235/54C07C311/13C07C311/20C07C2101/16
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Quick Facts
Patent No.
US 9,932,302
App. No.
14/519,679
Granted
Apr 3, 2018
Kind
B1
Abstract

The present disclosure provides compounds, compositions, and methods for use of the compounds. The compounds are N-phenyl or N-benzyl enaminones. The compositions can be pharmaceutical compositions. For example, the compounds/compositions are used in treating seizure disorders. The methods entail administering a composition comprising one or more of the compounds to a subject in need thereof. Articles of manufacture comprising one or more of the compounds/compositions are also provided.

Claims (13)

1. A compound having the following structure:

2. The compound of claim 1 , wherein the compound has the following structure:

3. A composition comprising a compound of claim 1 and a pharmaceutically acceptable carrier.

4. A method for treating a seizure in an individual in need thereof comprising administering to the individual a composition comprising a therapeutically effective amount of a compound of claim 1 .

5. The method of claim 4 , wherein the seizure is an epileptic seizure.

6. The method of claim 4 , wherein the seizure is a partial seizure.

7. The method of claim 4 , wherein the seizure is a generalized seizure.

8. The method of claim 4 , wherein the individual in need has previously experienced an epileptic seizure.

9. An article of manufacture comprising packaging and at least one container, wherein the container contains a composition comprising a compound of claim 1 , the article further comprising printed material, the printed material providing an indication that the composition is for use in treatment of a seizure disorder.

10. The article of claim 9 , wherein the seizure disorder is epilepsy.

11. The article of claim 9 , wherein the seizure disorder comprises partial seizures.

12. The article of claim 9 , wherein the seizure disorder comprises generalized seizures.

13. The compound of claim 1 , wherein the compound is active in at least in therapy resistance psychomotor (6-Hz) model.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 23, 2015
From: HARPER, TAWES; JACKSON-AYOTUNDE, PATRICE
To: UNIVERSITY OF MARYLAND, EASTERN SHORE
Reel/Frame 035281/0259 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 20, 2015
From: HARPER, TAWES; JACKSON-AYOTUNDE, PATRICE
To: UNIVERSITY OF MARYLAND, COLLEGE PARK
Reel/Frame 035218/0800 →
Continuity (1)
Provisional Application 61893652 · Oct 21, 2013