IP Library Granted Patent US 10,053,430
Granted Patent B2
US 10,053,430 · App. 15/636,562 · Granted Aug 21, 2018

RAF kinase modulator compounds and methods of use thereof

Inventors: Sunny Abraham (San Diego, CA); Shripad S. Bhagwat (San Diego, CA); Brian T. Campbell (Burlington, NJ); Qi Chao (San Diego, CA); Raffaella Faraoni (San Diego, CA); Mark W. Holladay (San Diego, CA); Andiliy G. Lai (San Diego, CA); Martin W. Rowbottom (San Diego, CA); Eduardo Setti (San Mateo, CA); Kelly G. Sprankle (Vista, CA)
Assignee: AMBIT BIOSCIENCES CORP.
C07D239/88C07D261/14
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Quick Facts
Patent No.
US 10,053,430
App. No.
15/636,562
Granted
Aug 21, 2018
Kind
B2
Abstract

Compounds, compositions and methods are provided for modulating the activity of RAF kinases, including BRAF kinase and for the treatment, prevention, or amelioration of one or more symptoms of disease or disorder mediated by RAF kinases.

Claims (3)

1. A compound which is

or a salt thereof.

2. A method of preparing the compound of claim 1 , or a salt thereof, comprising allowing 5,5,5-trifluoro-4,4-dimethyl-3-oxopentanenitrile to react with hydroxylamine, or a salt thereof.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 13, 2017
From: ABRAHAM, SUNNY; BHAGWAT, SHRIPAD S.; CAMPBELL, BRIAN T.; CHAO, QI; FARAONI, RAFFAELLA; HOLLADAY, MARK W.; LAI, ANDILIY G.; ROWBOTTOM, MARTIN W.; SETTI, EDUARDO; SPRANKLE, KELLY G.
To: AMBIT BIOSCIENCES CORP.
Reel/Frame 043192/0569 →
Continuity (7)
Continuation 15074671 · Mar 18, 2016
Continuation 14605834 · Jan 26, 2015
Continuation 14048655 · Oct 8, 2013
Continuation 12933402
Provisional Application 61069763 · Mar 17, 2008
Provisional Application 61110508 · Oct 31, 2008
Related Publication 20170298029A1 · Oct 19, 2017