IP Library Granted Patent US 10,071,103
Granted Patent B2
US 10,071,103 · App. 15/115,143 · Granted Sep 11, 2018

Treatments for resistant acne

Inventors: Shiladitya Sengupta (Delhi, IN); Suresh Rameshlal Chawrai (Pune, IN); Shamik Ghosh (Delhi, IN); Sumana Ghosh (Delhi, IN); Nilu Jain (New Delhi, IN); Suresh Sadhasivam (Salem, IN); Richard Buchta (Melbourne, AU); Anamika Bhattacharyya (Delhi, IN)
Assignee: VYOME BIOSCIENNCES PVT. LTD.
A61K31/55A61K9/0014A61K31/192A61K31/4709A61K45/06A61K47/02A61K47/08A61K47/10A61K47/183A61K47/32A61K47/36A61K47/38C07D513/04
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Quick Facts
Patent No.
US 10,071,103
App. No.
15/115,143
Granted
Sep 11, 2018
Kind
B2
Abstract

The present disclosure relates generally to novel molecules, compositions, and formulations for treatment of bacterial infections in general and more specifically to bacterial infections with antibiotic resistant pathogens.

Claims (38)

1. A formulation, wherein the formulation comprises:

(i) 0.5 to 4 (% w/w) Besifloxacin.HCl (Equivalent to Besifloxacin);

(ii) 2 to 7 (% w/w) diethylene glycol monoethyl ether;

(iii) 0.1 (% w/w) Edetate disodium dehydrate (EDTA);

(iv) 2 to 10 (% w/w) glycerin;

(v) 0.9 to 1.75 (% w/w) hydroxyethyl cellulose;

(vi) 0 to 0.8 (% w/w) carbomer;

(vii) 0.3 to 0.7 (% w/w) phenoxyethanol;

(viii) 2 to 7 (% w/w) polyethylene glycol 400;

(ix) 0 to 0.5 (% w/w) sodium hyaluronate;

(x) sodium hydroxide; and

(xi) purified water.

2. The formulation of claim 1 , wherein the formulation further comprises adapalene.

3. The formulation of claim 1 , wherein the formulation further comprises a second anti-bacterial agent.

4. A formulation comprising:

(i) 1 to 4 (% w/w) Besifloxacin.HCl (Equivalent to Besifloxacin);

(ii) 5 (% w/w) diethylene glycol monoethyl ether;

(iii) 0.1 (% w/w) Edetate disodium dehydrate (EDTA);

(iv) 5 (% w/w) glycerin;

(v) 0.5 to 1.5 (% w/w) hydroxyethyl cellulose;

(vi) 0.3 to 1.2 (% w/w) carbomer;

(vii) 0.7 (% w/w) phenoxyethanol;

(viii) 5 (% w/w) polyethylene glycol 400;

(ix) 0 to 1 (% w/w) sodium hyaluronate;

(x) sodium hydroxide; and

(xi) purified water.

5. The formulation of claim 4 , wherein the formulation further comprises adapalene.

6. A method for treating a bacterial infection, comprising administering a therapeutic effective amount of a formulation of claim 1 to a subject in need thereof.

7. The method of claim 6 , wherein the bacterial infection is by an antibiotic-resistant bacterial strain.

8. The method of claim 6 , wherein bacterial infection is by P. acnes.

9. The method of claim 8 , wherein P. acnes is a drug resistant strain.

10. The method of claim 9 , wherein the drug resistant acne is not responding to a therapeutic amount of clindamycin, minocycline, doxycycline, tetracycline or erythromycin.

11. A method for treating a bacterial infection, comprising administering a therapeutic effective amount of a formulation of claim 4 to a subject in need thereof.

12. The method of claim 11 , wherein the bacterial infection is by an antibiotic-resistant bacterial strain.

13. The method of claim 11 , wherein bacterial infection is by P. acnes.

14. The method of claim 13 , wherein P. acnes is a drug resistant strain.

15. The method of claim 14 , wherein the drug resistant stain is not responding to a therapeutic amount of at least one of clindamycin, minocycline, doxycycline, tetracycline and erythromycin.

16. The formulation of claim 4 , wherein the formulation further comprises a second anti-bacterial agent.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 3, 2019
From: VYOME BIOSCIENCES PRIVATE LIMITED
To: VYOME THERAPEUTICS LIMITED
Reel/Frame 047894/0134 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 30, 2017
From: SENGUPTA, SHILADITYA; CHAWRAI, SURESH RAMESHLAL; GHOSH, SHAMIK; GHOSH, SUMANA; JAIN, NILU; SADHASIVAM, SURESH; BUCHTA, RICHARD; BHATTACHARYYA, ANAMIKA
To: VYOME BIOSCIENCES PRIVATE LIMITED
Reel/Frame 042531/0267 →
Priority Claims (2)
IN 269/DEL/2014 · Jan 29, 2014 · national
IN 3247/DEL/2014 · Nov 10, 2014 · national
Continuity (1)
Related Publication 20160346294A1 · Dec 1, 2016
Cited By (5)
US 12,194,124 US 12,201,713 US 12,251,584 US 12,409,211 US 12,458,613