IP Library Granted Patent US 10,172,860
Granted Patent B2
US 10,172,860 · App. 15/659,526 · Granted Jan 8, 2019

Modulators of toll-like receptors

Inventors: Manoj C. Desai (Pleasant Hill, CA); Randall L. Halcomb (Foster City, CA); Paul Hrvatin (South San Francisco, CA); Hon Chung Hui (San Mateo, CA); Ryan McFadden (Foster City, CA); Paul A. Roethle (San Francisco, CA); Hong Yang (Fremont, CA)
Assignee: GILEAD SCIENCES, INC.
A61K31/519A61K31/527A61K31/5377A61K31/551A61K31/573A61K31/683A61K31/708A61K31/7056A61K31/7072A61K38/16A61K38/21A61K38/212A61K45/06C07D403/12C07D475/06C07D475/08C07D475/10C07D475/12C07D487/04Y02A50/385Y02A50/387Y02A50/389Y02A50/391Y02A50/393Y02A50/395
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Quick Facts
Patent No.
US 10,172,860
App. No.
15/659,526
Granted
Jan 8, 2019
Kind
B2
Abstract

Provided are modulators of TLRs of Formula II: pharmaceutically acceptable salts thereof, compositions containing such compounds, and therapeutic methods that include the administration of such compounds.

Claims (23)

1. A compound of the Formula:

or a pharmaceutically acceptable salt thereof, wherein:

L 1 is —O—, —S—, —S(O) 2 —, or —S(O)—;

R 1 is alkyl;

X 1 is alkylene;

D is phenyl;

L 2 is alkylene;

n is 0;

R 4 and R 5 are each independently H; and

R 6 and R 7 , taken together with the nitrogen to which they are both attached, form an unsubstituted 4-6 membered heterocycle, which may contain one or more additional heteroatoms selected from N, O, or S.

2. The compound of claim 1 , wherein L 1 is —O—.

3. The compound of claim 1 , wherein X 1 is —CH 2 —.

4. The compound of claim 1 , wherein L 2 is —CH 2 —.

5. The compound of claim 1 , selected from the group consisting of:

or a salt thereof.

6. The compound of claim 1 , selected from the group consisting of:

or a salt thereof.

7. The compound of claim 1 , selected from the group consisting of:

or a salt thereof.

8. The compound of claim 1 , selected from the group consisting of:

or a salt thereof.

9. The compound of claim 1 , having the structure:

or a salt thereof.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 11, 2017
From: DESAI, MANOJ C.; HALCOMB, RANDALL L.; HRVATIN, PAUL; HUI, HON CHUNG; MCFADDEN, RYAN; ROETHLE, PAUL A.; YANG, HONG
To: GILEAD SCIENCES, INC.
Reel/Frame 043548/0783 →
Continuity (12)
Continuation 15244943 · Aug 23, 2016
Continuation 14804145 · Jul 20, 2015
Continuation 14321689 · Jul 1, 2014
Continuation 14089633 · Nov 25, 2013
Continuation 13679803 · Nov 16, 2012
Continuation 12632194 · Dec 7, 2009
Provisional Application 61242635 · Sep 15, 2009
Provisional Application 61227378 · Jul 21, 2009
Provisional Application 61224386 · Jul 9, 2009
Provisional Application 61170404 · Apr 17, 2009
Provisional Application 61121061 · Dec 9, 2008
Related Publication 20180085370A1 · Mar 29, 2018
Cited By (4)
US 12,311,010 US 12,486,271 US 12,611,453 US 12,702,695