IP Library Granted Patent US 10,201,558
Granted Patent B2
US 10,201,558 · App. 14/855,065 · Granted Feb 12, 2019

Compositions of selenoorganic compounds and methods of use thereof

Inventors: Ronan Power (Lexington, KY); Zi-Jian Lan (Lexington, KY)
Assignee: Alltech, Inc.
A61K31/7135A61K31/28A61K31/7076A61K38/05A61K38/28C07D473/34A61K31/706A61K31/7064
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,201,558
App. No.
14/855,065
Granted
Feb 12, 2019
Kind
B2
Abstract

The present application relates to compositions comprising selenium compounds, such as 5′-Methylselenoadenosine, a compound of Formula (I), and combinations thereof, and methods of using the same for inhibiting β amyloid aggregation, ApoE4 expression, p38 or Tau protein phosphorylation, or increasing Neprilysin and Insulin Degrading Enzyme expression.

Claims (16)

1. A method for inhibiting β amyloid aggregation in a subject in need thereof comprising:

administering a composition to a subject, the composition comprising at least 0.1% (w/v) of 5′-deoxy-5′-methylselenoadenosine, or a pharmaceutically acceptable salt thereof; and a carrier.

2. A method for inhibiting ApoE4 expression in a subject in need thereof comprising:

administering a composition to a subject, the composition comprising at least 0.1% (w/v) of 5′-deoxy-5′-methylselenoadenosine, or a pharmaceutically acceptable salt thereof; and a carrier.

3. A method of decreasing p38 phosphorylation in a subject in need thereof comprising:

administering a composition to a subject, the composition comprising at least 0.1% (w/v) of 5′-deoxy-5′-methylselenoadenosine, or a pharmaceutically acceptable salt thereof; and a carrier.

4. A method of increasing neprilysin expression in a subject in need thereof comprising:

administering a composition to a subject, the composition comprising at least 0.1% (w/v) of 5′-deoxy-5′-methylselenoadenosine, or a pharmaceutically acceptable salt thereof; and a carrier.

5. A method of decreasing beta-secretase (BACE) expression in a subject in need thereof comprising:

administering a composition to a subject, the composition comprising at least 0.1% (w/v) of 5′-deoxy-5′-methylselenoadenosine, or a pharmaceutically acceptable salt thereof; and a carrier.

6. A method of increasing insulin-degrading enzyme (IDE) expression in a subject in need thereof comprising:

administering a composition to a subject, the composition comprising at least 0.1% (w/v) of 5′-deoxy-5′-methylselenoadenosine, or a pharmaceutically acceptable salt thereof; and a carrier.

7. A method for inhibiting β amyloid aggregation in a subject in need thereof comprising:

administering a composition to a subject, the composition comprising at least 0.033% (w/v) of 5′-deoxy-5′-methylselenoadenosine, or a pharmaceutically acceptable salt thereof; and a carrier.

8. A method of decreasing phosphorylated tau (pTau) expression in a subject in need thereof comprising:

administering a composition to a subject, the composition comprising at least 0.1% (w/v) of 5′-deoxy-5′-methylselenoadenosine, or a pharmaceutically acceptable salt thereof; and a carrier.

Assignments (7)
SECOND LIEN PATENT SECURITY AGREEMENT Recorded Nov 14, 2024
From: ALLTECH, INC.; RIDLEY USA INC.
To: WILMINGTON TRUST, NATIONAL ASSOCIATION, AS ADMINISTRATIVE AGENT
Reel/Frame 069357/0281 →
PATENT SECURITY AGREEMENT Recorded Dec 1, 2021
From: ALLTECH, INC.
To: BANK OF AMERICA, N.A., AS ADMINISTRATIVE AGENT
Reel/Frame 058292/0934 →
TERMINATION AND RELEASE OF SECURITY INTEREST IN PATENTS (2) Recorded Nov 30, 2021
From: BANK OF AMERICA, N.A., AS ADMINISTRATIVE AGENT
To: ALLTECH, INC.
Reel/Frame 058282/0440 →
RELEASE OF SECURITY INTEREST Recorded Oct 26, 2021
From: WILMINGTON TRUST, NATIONAL ASSOCIATION, AS ADMINISTRATIVE AGENT
To: ALLTECH, INC.; RIDLEY USA INC.
Reel/Frame 057919/0761 →
ASSIGNMENT FOR SECURITY -- PATENTS Recorded May 18, 2020
From: ALLTECH, INC; RIDLEY USA, INC
To: WILMINGTON TRUST, NATIONAL ASSOCIATION, AS ADMINISTRATIVE AGENT
Reel/Frame 052694/0412 →
PATENT SECURITY AGREEMENT Recorded Apr 19, 2016
From: ALLTECH, INC.
To: BANK OF AMERICA, N.A., AS ADMINISTRATIVE AGENT
Reel/Frame 038464/0013 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 17, 2015
From: POWER, RONAN; LAN, ZI-JIAN
To: ALLTECH, INC.
Reel/Frame 036594/0354 →
Continuity (2)
Continuation In Part PCTUS2014029542 · Mar 14, 2014
Related Publication 20160082033A1 · Mar 24, 2016