IP Library Granted Patent US 10,456,439
Granted Patent B2
US 10,456,439 · App. 15/518,553 · Granted Oct 29, 2019

NK3 agonist for use in the treatment of a patient suffering from atrial arrhythmia or fibrillation

Inventors: Ruben Coronel (Abcoude, NL); Marieke Veldkamp (Leiden, NL)
Assignee: Academisch Medisch Centrum
A61K38/046A61K9/0019A61K9/0053
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Quick Facts
Patent No.
US 10,456,439
App. No.
15/518,553
Granted
Oct 29, 2019
Kind
B2
Abstract

The invention relates to an NK3 agonist or a pharmaceutically acceptable salt or solvate thereof, for use in the treatment of a atrial arrhythmia. The invention further relates to a composition comprising an NK3 agonist for use in the treatment of a patient suffering from a disease wherein the electrical activity of an atrial heart cell is affected.

Claims (20)

1. A method for treating atrial arrhythmia comprising administering to a subject in need thereof an NK3 agonist selected from the group consisting of Neurokinin B (NKB), Neurokinin A (NKA), Hemokinin 1 (HEK1), Eledoisin, Kassinin, Senktide [succinyl-(Asp6, MePhe8)-SP(6-11)], [MePhe7]-NKB (1a), Pro7-NKB, and a pharmaceutically acceptable salt thereof.

2. The method according to claim 1 , wherein said NK3 agonist is selected from the group consisting of Neurokinin B (NKB), Pro7-NKB, Neurokinin A (NKA) and Senktide.

3. The method according to claim 1 , wherein said NK3 agonist is formulated in a composition comprising a pharmaceutically acceptable carrier.

4. The method according to claim 3 , wherein said composition is formulated for intravenous administration.

5. The method according to claim 4 , wherein said NK3 agonist is selected from the group consisting of Neurokinin B (NKB), Pro7-NKB, Neurokinin A (NKA) and Senktide.

6. The method according to claim 3 , wherein said composition is formulated for oral administration.

7. The method according to claim 6 , wherein the NK3 agonist is selected from the group consisting of Neurokinin B (NKB), Pro7-NKB, Neurokinin A (NKA) and Senktide.

8. The method according to claim 3 , wherein said NK3 agonist is selected from the group consisting of Neurokinin B (NKB), Pro7-NKB, Neurokinin A (NKA) and Senktide.

9. The method according to claim 3 , wherein said subject is a human.

10. The method according to claim 3 , wherein said NK3 agonist is Neurokinin B (NKB).

11. The method according to claim 3 , wherein said NK3 agonist is Pro7-NKB.

12. The method according to claim 3 , wherein said NK3 agonist is Neurokinin A (NKA).

13. The method according to claim 3 , wherein said NK3 agonist is Senktide.

14. The method according to claim 3 , wherein said NK3 agonist is Neurokinin B (NKB), Pro7-NKB, Neurokinin A (NKA) and Senktide.

15. The method according to claim 3 , further comprising administering one or more additional therapeutic agent to the subject.

16. The method according to claim 15 , wherein the one or more additional therapeutic agent is selected from the group consisting of digoxin, beta blockers, amiodarone, disopyramide, calcium antagonists, Sotalol, flecanaide, procainamide, quinidine and propafenone.

17. The method according to claim 15 , wherein the NK3 agonist and the one or more additional therapeutic agent are administered simultaneously.

18. The method according to claim 15 , comprising administering sequentially to the subject the NK3 agonist, followed by the one or more additional therapeutic agent.

19. The method according to claim 15 , comprising administering sequentially to the subject the one or more additional therapeutic agent, followed by the NK3 agonist.

20. A method for treating a disease caused by abnormal electrical conduction in the atrial muscle tissue of a subject, comprising administering to the subject an NK3 agonist selected from the group consisting of Neurokinin B (NKB), Neurokinin A (NKA), Hemokinin 1 (HEK1), Eledoisin, Kassinin, Senktide [succinyl-(Asp6, MePhe8)-SP(6-11)], [MePhe7]-NKB (1a), Pro7-NKB, and a pharmaceutically acceptable salt thereof.

Assignments (2)
CHANGE OF NAME Recorded Sep 11, 2024
From: ACADEMISCH MEDISCH CENTRUM
To: STICHTING AMSTERDAM UMC
Reel/Frame 068942/0762 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2017
From: CORONEL, RUBEN; VELDKAMP, MARIEKE
To: ACADEMISCH MEDISCH CENTRUM
Reel/Frame 042481/0891 →
Priority Claims (1)
EP 14189212 · Oct 16, 2014 · regional
Continuity (1)
Related Publication 20190015471A1 · Jan 17, 2019