IP Library Granted Patent US 11,090,293
Granted Patent B2
US 11,090,293 · App. 16/998,295 · Granted Aug 17, 2021

Use of gaboxadol for the treatment of Tourette syndrome, tics and stuttering

Inventor: Matthew During (Weston, CT)
Assignee: Ovid Therapeutics Inc.
A61K31/437A61P25/14
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Quick Facts
Patent No.
US 11,090,293
App. No.
16/998,295
Granted
Aug 17, 2021
Kind
B2
Abstract

Treatment of Tourette syndrome using gaboxadol or a pharmaceutically acceptable salt thereof is provided. Treatment of tics using gaboxadol or a pharmaceutically acceptable salt thereof is provided. Treatment of stuttering using gaboxadol or a pharmaceutically acceptable salt thereof is provided. Therapeutic compositions that may be used to improve one or more symptoms of Tourette syndrome are provided. Therapeutic compositions that may be used to improve one or more symptoms of tics are provided. Also provided are therapeutic compositions that may be used to improve one or more symptoms of stuttering.

Claims (11)

1. A method of treating stuttering comprising administering to a patient in need thereof about 0.05 mg to about 30 mg gaboxadol or a pharmaceutically acceptable salt thereof, wherein the method provides improvement in one or more symptoms of the stuttering in the patient.

2. The method of claim 1 , wherein the improvement is provided for more than 6 hours after administration.

3. The method of claim 1 , wherein the patient is administered a composition comprising about 1 mg to about 15 mg gaboxadol or a pharmaceutically acceptable salt thereof.

4. The method of claim 1 , wherein the in vivo plasma profile of the patient 6 hours after administration of the gaboxadol or pharmaceutically acceptable salt thereof is reduced by more than 50%.

5. The method of claim 1 , wherein the AUC 6-12 of the patient 6 hours after administration of the gaboxadol or pharmaceutically acceptable salt thereof is less than 75% of the administered dose.

6. The method of claim 1 , wherein the method provides improvement in at least one symptom selected from the group consisting of repetition of sounds, repetition of syllables, repetition of words, prolongation of sounds, blocks and struggle behaviors.

7. The method of claim 1 , wherein the method provides improvement in the patient for at least 12 hours.

8. The method of claim 1 , wherein the stuttering is developmental stuttering.

9. The method of claim 1 , wherein the stuttering is neurogenic stuttering.

10. A method of treating stuttering comprising administering to a patient in need thereof gaboxadol or a pharmaceutically acceptable salt thereof wherein the method provides an in vivo plasma profile comprising a C max less than about 400 ng/ml and wherein the method provides improvement in the patient for more than 6 hours after administration of the gaboxadol or a pharmaceutically acceptable salt thereof.

11. A method of treating stuttering comprising administering to a patient in need thereof gaboxadol or a pharmaceutically acceptable salt thereof wherein the method provides an in vivo plasma profile comprising a AUC 6-12 of less than about 900 ng·hr/ml and wherein the method provides improvement in the patient for more than 6 hours after administration of the gaboxadol or a pharmaceutically acceptable salt thereof.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 20, 2020
From: DURING, MATTHEW
To: OVID THERAPEUTICS INC.
Reel/Frame 053552/0079 →
Continuity (3)
Continuation 16577084 · Sep 20, 2019
Provisional Application 62733730 · Sep 20, 2018
Related Publication 20200375960A1 · Dec 3, 2020