IP Library › Granted Patent US 11,655,257
Granted Patent B2
US 11,655,257 · App. 17/148,903 · Granted May 23, 2023

MK2 inhibitors, synthesis thereof, and intermediates thereto

Inventors: Gregg Brian Feigelson (Chester, NY); Maryll E. Geherty (Pennington, NJ); Richard Martin Heid, Jr. (Maplewood, NJ); Mohit Kothare (Bridgewater, NJ); Hon-Wah Man (Princeton, NJ); Alexander L. Ruchelman (Cream Ridge, NJ); John F. Traverse (Lebanon, NJ); Kelvin Hin-Yeong Yong (Westfield, NJ); Chengmin Zhang (Florham Park, NJ)
Assignee: Celgene CAR LLC
C07D495/14
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Quick Facts
Patent No.
US 11,655,257
App. No.
17/148,903
Granted
May 23, 2023
Kind
B2
Abstract

The present invention provides methods of preparing a MK2 inhibitor, and intermediates related thereto.

Claims (21)

1. A compound selected from the group consisting of:

or a salt thereof.

2. The compound of claim 1 , selected from the group consisting of:

or a salt thereof.

3. The compound of claim 2 , wherein the compound is:

or a salt thereof.

4. The compound of claim 2 , wherein the compound is:

or a salt thereof.

5. The compound of claim 2 , wherein the compound is:

or a salt thereof.

6. The compound of claim 2 , wherein the compound is:

or a salt thereof.

7. The compound of claim 2 , wherein the compound is:

or a salt thereof.

8. The compound of claim 1 , selected from the group consisting of:

and

and or a salt thereof.

9. The compound of claim 8 , wherein the compound is:

or a salt thereof.

10. The compound of claim 8 , wherein the compound is:

or a salt thereof.

Assignments (2)
NUNC PRO TUNC ASSIGNMENT Recorded May 3, 2023
From: CELGENE CAR LLC
To: BRISTOL-MYERS SQUIBB COMPANY
Reel/Frame 063526/0959 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 14, 2021
From: FEIGELSON, GREGG BRIAN; GEHERTY, MARYLL E.; HEID, RICHARD MARTIN, JR.; KOTHARE, MOHIT; MAN, HON-WAH; RUCHELMAN, ALEXANDER L.; TRAVERSE, JOHN F.; YONG, KELVIN HIN-YEONG; ZHANG, CHENGMIN
To: CELGENE CAR LLC
Reel/Frame 055912/0555 →
Continuity (3)
Division 16494701
Provisional Application 62472024 · Mar 16, 2017
Related Publication 20210139501A1 · May 13, 2021