IP Library Granted Patent US 11,957,749
Granted Patent B2
US 11,957,749 · App. 16/772,194 · Granted Apr 16, 2024

Hepatitis B immunization regimen and compositions

Inventors: Virginia Ammendola (Rome, IT); Babak Bayat (Rixensart, BE); Clarisse Lorin (Rixensart, BE); Ventzislav Bojidarov Vassilev (Rixensart, BE); Alessandra Vitelli (Rome, IT)
Assignee: GlaxoSmithKline Biologicals SA
A61K39/292A61K39/39A61P31/20C07K14/005C12N7/00A61K2039/5254A61K2039/5256A61K2039/55555A61K2039/55572A61K2039/55577A61K2039/57C07K2319/40C12N2710/10343C12N2710/24143C12N2730/10122C12N2730/10134
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Quick Facts
Patent No.
US 11,957,749
App. No.
16/772,194
Granted
Apr 16, 2024
Kind
B2
Abstract

The present invention relates to immunogenic compositions and combinations thereof which may find use in immunisation regimens for the treatment of chronic hepatitis B. An immunogenic composition comprises a replication-defective chimpanzee adenoviral (ChAd) vector comprising polynucleotides encoding HBs, HBc human invariant chain (hIi) fused to the HBc. Another immunogenic composition comprises a Modified Vaccinia Virus Ankara (MVA) vector comprising polynucleotides encoding HBs and HBc. Another immunogenic composition comprises recombinant HBs, C-terminal truncated recombinant HBc and an adjuvant containing MPL and QS-21.

Claims (16)

1. An immunogenic composition comprising a Modified Vaccinia Virus Ankara (MVA) vector comprising a polynucleotide encoding a hepatitis B surface antigen (HBs) and a polynucleotide encoding a hepatitis B virus core antigen (HBc), wherein the polynucleotides encoding HBs and HBc are separated by a polynucleotide encoding the 2A cleaving region of the foot and mouth disease virus (FMDV).

2. An immunogenic composition comprising a recombinant hepatitis B surface antigen (HBs), a C-terminal truncated recombinant hepatitis B virus core antigen (HBc), and an adjuvant containing MPL and QS-21; wherein the ratio of recombinant HBc to recombinant HBs in the composition is about 1.5:1, 2:1, 2.5:1, 3:1, 3.5:1, 4:1, 4.5:1, 5:1, 5.5:1, or 6:1.

3. An immunogenic combination comprising:

a) a composition comprising a replication-defective chimpanzee adenoviral (ChAd) vector comprising a polynucleotide encoding a hepatitis B surface antigen (HBs) and a polynucleotide encoding a hepatitis B virus core antigen (HBc);

b) a composition comprising a Modified Vaccinia Virus Ankara (MVA) vector comprising a polynucleotide encoding a hepatitis B surface antigen (HBs) and a polynucleotide encoding a hepatitis B virus core antigen (HBc), wherein the polynucleotides encoding HBs and HBc are separated by a polynucleotide encoding the 2A cleaving region of the foot and mouth disease virus (FMDV); and

c) a composition comprising a recombinant hepatitis B surface antigen (HBs), a recombinant hepatitis B virus core antigen (HBc) comprising amino acids 1-145, 1-146, 1-147, 1-148, or 1-149 of a wild-type hepatitis B virus core antigen protein, and an adjuvant.

4. The immunogenic combination according to claim 3 , wherein the ChAd vector of component a) of the combination further comprises a polynucleotide encoding the human invariant chain (hli) fused to the HBc, the recombinant HBc of component c) of the combination is C-terminal truncated, the adjuvant of component c) of the combination contains MPL and QS-21, and the ratio of recombinant HBc to recombinant HBs of component c) of the combination is about 1.5:1, 2:1, 2.5:1, 3:1, 3.5:1, 4:1, 4.5:1, 5:1, 5.5:1, or 6:1.

5. A kit comprising the following components:

a) a composition comprising a replication-defective chimpanzee adenoviral (ChAd) vector comprising a polynucleotide encoding a hepatitis B surface antigen (HBs) and a polynucleotide encoding a hepatitis B virus core antigen (HBc);

b) a composition comprising a Modified Vaccinia Virus Ankara (MVA) vector comprising a polynucleotide encoding a hepatitis B surface antigen (HBs) and a polynucleotide a hepatitis B virus core antigen (HBc), wherein the polynucleotides encoding HBs and HBc are separated by a polynucleotide encoding the 2A cleaving region of the foot and mouth disease virus (FMDV); and

c) a composition comprising a recombinant hepatitis B surface antigen (HBs), a recombinant hepatitis B virus core antigen (HBc) comprising amino acids 1-145, 1-146, 1-147, 1-148, or 1-149 of a wild-type hepatitis B core antigen protein, and an adjuvant,

with instructions for administration of the components sequentially or concomitantly for the treatment of chronic hepatitis B (CHB).

6. The immunogenic combination according to claim 3 , wherein the HBc of component b) comprises SEQ ID NO:11 or an amino acid sequence at least 98% homologous thereto and the HBs of component b) comprises SEQ ID NO:1 or an amino acid sequence at least 98% homologous thereto, wherein the polynucleotides encoding the HBc and HBs of component b) are separated by a polynucleotide encoding an amino acid sequence comprising SEQ ID NO:3, or an amino acid sequence at least 98% homologous thereto.

7. The immunogenic combination according to claim 3 , wherein the MVA vector of component b) comprises a polynucleotide encoding the amino acid sequence of SEQ ID NO:5.

8. The immunogenic combination according to claim 3 , wherein the MVA vector of component b) comprises a polynucleotide having the nucleotide sequence of SEQ ID NO:6.

9. The immunogenic combination according to claim 3 , wherein the composition of component c) comprises a recombinant HBs (SEQ ID NO:1), a recombinant HBc comprising amino acids 1-149 (SEQ ID NO:2) and an adjuvant comprising MPL, QS-21 and liposomes composed of dioleoyl phosphatidylcholine (DOPC) and cholesterol in a phosphate buffered saline solution.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 7, 2024
From: BAYAT, BABAK; LORIN, CLARISSE; VASSILEV, VENTZISLAV BOJIDAROV
To: GLAXOSMITHKLINE BIOLOGICALS SA
Reel/Frame 066687/0293 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 16, 2024
From: VITELLLI, ALESSANDRA; AMMENDOLA, VIRGINIA; REITHERA SRL
To: GLAXOSMITHKLINE BIOLOGICALS SA
Reel/Frame 066134/0346 →
Priority Claims (1)
GB 1721069 · Dec 15, 2017 · national
Continuity (1)
Related Publication 20210154290A1 · May 27, 2021