IP Library Granted Patent US 12,138,249
Granted Patent B2
US 12,138,249 · App. 18/118,012 · Granted Nov 12, 2024

Compositions and methods for treating conditions related to elevated levels of eosinophils and/or basophils

Inventors: Michael E. Bozik (Pittsburgh, PA); Gregory Hebrank (Greensburg, PA); Wildon Farwell (Wayland, MA); Thomas Petzinger, Jr. (Pittsburgh, PA); Steven Dworetzky (Jefferson Hills, PA)
Assignee: Areteia Therapeutics, Inc.
A61K31/428A61K45/06Y02A50/30
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Quick Facts
Patent No.
US 12,138,249
App. No.
18/118,012
Granted
Nov 12, 2024
Kind
B2
Abstract

Disclosed herein are methods of treating conditions, which may be associated with elevated levels of eosinophils and/or basophils, with a therapeutically effective amount of dexpramipexole or pharmaceutical acceptable salt thereof.

Claims (15)

1. A method of treating a condition characterized by increased numbers of eosinophils in a subject comprising:

administering to a subject in need thereof a therapeutically effective amount of R(+) pramipexole, or a pharmaceutically acceptable salt thereof, wherein the condition is a gastrointestinal disease.

2. The method of claim 1 , wherein the condition is characterized by eosinophil numbers above about 100 cells per microliter in the peripheral blood.

3. The method of claim 1 , wherein the therapeutically effective amount of R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is from about 50 mg to about 1,500 mg per day.

4. The method of claim 1 , wherein the therapeutically effective amount of R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is from about 150 mg to about 1,500 mg per day.

5. The method of claim 1 , wherein the therapeutically effective amount of R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is from about 150 mg to about 300 mg per day.

6. The method of claim 1 , wherein the therapeutically effective amount of R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is about 150 mg per day.

7. The method of claim 1 , wherein the therapeutically effective amount of R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is about 300 mg per day.

8. The method of claim 1 , wherein R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is administered two or more times per day.

9. The method of claim 1 , wherein R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is administered at a fraction of a daily dose two or more times per day.

10. The method of claim 8 , wherein R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is administered two times per day.

11. The method of claim 10 , wherein the dose is administered every 12 hours.

12. The method of claim 1 , wherein R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is administered at about 150 mg two times per day.

13. The method of claim 1 , further comprising administering a second therapeutic agent that is capable of decreasing eosinophil levels, the agent selected from the group consisting of a glucocorticoid, a corticosteroid, a non-steroidal anti-inflammatory drug (NSAID), a tyrosine kinase inhibitor, a fusion protein, a monoclonal antibody directed against one or more pro-inflammatory cytokines, a chemotherapeutic agent and a combination thereof.

14. The method of claim 1 , wherein R(+) pramipexole, or a pharmaceutically acceptable salt thereof, is administered orally.

Assignments (6)
RELEASE OF SECURITY INTEREST Recorded Nov 21, 2025
From: HERCULES CAPITAL, INC., AS AGENT
To: ARETEIA THERAPEUTICS, INC.
Reel/Frame 072993/0621 →
SECURITY INTEREST Recorded Oct 10, 2025
From: ARETEIA THERAPEUTICS, INC.
To: HERCULES CAPITAL, INC., AS AGENT
Reel/Frame 072540/0980 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2023
From: KNOPP BIOSCIENCES LLC
To: ARETEIA THERAPEUTICS, INC.
Reel/Frame 063727/0581 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2023
From: BOZIK, MICHAEL E.; HEBRANK, GREGORY; DWORETZKY, STEVEN; PETZINGER, THOMAS, JR.
To: KNOPP BIOSCIENCES LLC
Reel/Frame 063727/0695 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2023
From: FARWELL, WILDON
To: BIOGEN MA, INC.
Reel/Frame 063727/0825 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2023
From: BIOGEN MA, INC.
To: KNOPP BIOSCIENCES LLC
Reel/Frame 063727/0891 →
Continuity (9)
Continuation 16950973 · Nov 18, 2020
Continuation 15923650 · Mar 16, 2018
Continuation 14904058
Continuation In Part PCTUS2013054804 · Aug 13, 2013
Continuation In Part 13966229 · Aug 13, 2013
Provisional Application 61859158 · Jul 26, 2013
Provisional Application 61845944 · Jul 12, 2013
Provisional Application 61865118 · Aug 12, 2013
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