IP Library Granted Patent US 12,331,027
Granted Patent B2
US 12,331,027 · App. 16/763,004 · Granted Jun 17, 2025

Herbicidal pyridylethers

Inventors: Manuel Johannes (Duesseldorf, DE); Laetitia Souillart (Ludwigshafen, DE); Matthias Witschel (Ludwigshafen, DE); Tobias Seiser (Limburgerhof, DE); Liliana Parra Rapado (Limburgerhof, DE); Raphael Aponte (Limburgerhof, DE); Thomas Mietzner (Ludwigshafen, DE); Trevor William Newton (Limburgerhof, DE); Thomas Seitz (Ludwigshafen, DE); Peter Dombo (Limburgerhof, DE)
C07D401/04A01N43/40A01N43/54A01N43/56A01N43/58A01N43/653A01N43/66A01N43/82C07D213/73C07D213/74C07D401/12C07D401/14C07D413/04C07D471/04
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Quick Facts
Patent No.
US 12,331,027
App. No.
16/763,004
Granted
Jun 17, 2025
Kind
B2
Abstract

The present invention relates to pyridylethers of formula (I) or their agriculturally acceptable salts or derivatives, wherein the variables are defined accord-ing to the description, processes and intermediates for preparing the pyridylethers of formula (I), compositions comprising them and their use as herbicides, i.e. for controlling harmful plants, and also a method for controlling unwanted vegetation which comprises allowing a herbicidal effective amount of at least one pyridylether of formula (I) to act on plants, their seed and/or their habitat.

Claims (40)

1. A pyridylether of formula (I)

wherein the variables have the following meanings:

R 1 is H or halogen;

R 2 is H, halogen;

R 3 is H;

R 4 is H;

R 5 is OR 6 , wherein

R 6 is hydrogen, C 1 -C 6 -alkyl

n is 1;

Q is O;

W is O;

X is O;

Y is a heterocycle selected from the group consisting of Y 2 , Y 13 , Y 31 , Y 37 , Y 38 , Y 39 , or Y 67

wherein

A 1 , A 2 , A 3 are oxygen or sulphur;

A 4 is sulphur;

R 19 , R 21 , R 22 , R 23 , R 24 are hydrogen, C 1 -C 6 -haloalkyl, or C 1 -C 6 -haloalkyl; or

R 21 and R 22 together with the atoms to which they are attached, form a five- or six-membered cycle, which is saturated or partially unsaturated, which may comprise apart from carbon atoms one to two nitrogen atoms, and which for its part may be partially or fully halogenated, and which for its part may be substituted by one to two C 1 -C 6 -alkyl radicals;

R 26 and R 27 are C 1 -C 6 -alkyl;

R 28 is halogen or C 1 -C 6 -alkyl;

R 35 and R 36 are C 1 -C 6 -alkyl;

Z is Z-1 or Z-7

wherein

* denotes the point of attachment of Z to X;

* denotes the point of attachment of Z to Q; and

R a , R b , R c , and R d are H,

or an agriculturally salt thereof.

2. The pyridylether of formula (I) according to claim 1 wherein R 1 is H or F, and R 2 is F, or Cl.

3. A process for the preparation of a pyridylether of formula (I) as defined in claim 1 , comprising reacting pyridines of formula (II)

wherein R 1 , R 2 and Y are as defined in claim 1 ; and

L 1 is halogen, C 1 -C 6 -alkylsulfonate or arylsulfonate;

with compounds of formula (III)

wherein R 3 , R 4 , R 5 , n, Q, W, X and Z are as defined in claim 1 ;

in the presence of a base.

4. A herbicidal composition comprising an herbicidally active amount of at least one pyridylether of formula (I) as claimed in claim 1 and at least one inert liquid and/or solid carrier and, optionally, at least one surface-active substance.

5. A process for the preparation of herbicidal active compositions, which comprises mixing an herbicidally active amount of at least one pyridylether of formula (I) as claimed in claim 1 and at least one inert liquid and/or solid carrier and, optionally, at least one surface-active substance.

6. A method of controlling undesired vegetation, which comprises applying an herbicidally active amount of at least one pyridylether of formula (I) as claimed in claim 1 to the undesired vegetation, the environment thereof, or seed thereof.

7. A pyridylether of formula (I) as claimed in claim 1 for use as an herbicide.

8. The pyridylether of formula (I) according to claim 2 wherein R 1 is H and R 2 is F or Cl.

9. The pyridylether of formula (I) according to claim 2 wherein R 1 is F and R 2 is F or Cl.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 12, 2020
From: JOHANNES, MANUEL; SOUILLART, LAETITIA; WITSCHEL, MATTHIAS; SEISER, TOBIAS; PARRA RAPADO, LILIANA; APONTE, RAPHAEL; MIETZNER, THOMAS; NEWTON, TREVOR WILLIAM; SEITZ, THOMAS; DOMBO, PETER
To: BASF SE
Reel/Frame 054347/0763 →
Priority Claims (2)
EP 17203280 · Nov 23, 2017 · regional
EP 18169740 · Apr 27, 2018 · regional
Continuity (1)
Related Publication 20200392103A1 · Dec 17, 2020
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