IP Library › Granted Patent US 8,288,339
Granted Patent B2
US 8,288,339 · App. 12/297,705 · Granted Oct 16, 2012

GLP-1 compounds

Assignee: Amgen Inc.
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Quick Facts
Patent No.
US 8,288,339
App. No.
12/297,705
Granted
Oct 16, 2012
Kind
B2
Abstract

GLP-1 compounds comprising GLP-1 analogs and methods of using the GLP-1 compounds for treating metabolic disorders, enhancing insulin expression, and promoting insulin secretion in a patient are provided.

Claims (7)

1. A GLP-1 compound comprising a GLP-1 analog that comprises the amino acid sequence of SEQ ID NO:18.

2. The GLP-1 compound of claim 1 , further comprising a water-soluble polymer.

3. The GLP-1 compound of claim 2 , wherein the water-soluble polymer is selected from the group consisting of polyethylene glycol, monomethoxy-polyethylene glycol, dextran, cellulose, poly-(N-vinyl pyrrolidone) polyethylene glycol, propylene glycol homopolymers, polypropylene oxide/ethylene oxide co-polymers, polyoxyethylated polyols, and polyvinyl alcohol.

4. A method for treating a subject with a metabolic disorder, comprising administering to the subject an effective amount of a GLP-1 compound of claim 1 , wherein the metabolic disorder is selected from the group of diabetes, impaired glucose tolerance, insulin resistance, irritable bowel syndrome, obesity and metabolic syndrome.

5. A method for treating a coronary disease or a lipid disorder in a subject, comprising administering to the subject a GLP-1 compound of claim 1 , wherein the coronary disease or lipid disorder is selected from the group consisting of hypertension, coronary artery disease, hyperlipidemia, cardiovascular disease, atherosclerosis, hypercholesteremia and myocardial infarction.

6. A method for treating a subject, comprising administering to the subject a GLP-1 compound of claim 1 , wherein the amount of the GLP administered is an amount sufficient to stimulate insulin release, reduce blood glucose levels, increase plasma insulin levels, increase beta-cell mass, induce satiety, reduce gastric secretion, delay gastric emptying or reduce gastric motility in the subject.

7. A pharmaceutical composition comprising the GLP-1 compound of claim 1 .

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 5, 2009
From: GEGG, COLIN VICTOR, JR; MIRANDA, LESLIE PHILLIP; WINTERS, KATHERINE ANN; VENIANT-ELLISON, MURIELLE
To: AMGEN INC.
Reel/Frame 022210/0532 →
Continuity (2)
Provisional Application 60793707 · Apr 20, 2006
Related Publication 20100048468A1 · Feb 25, 2010