IP Library › Granted Patent US 8,790,711
Granted Patent B2
US 8,790,711 · App. 13/624,856 · Granted Jul 29, 2014

Treating diabetes with a whole, leech saliva extract

Inventors: Abbas Mohammad Ghawi (Selangor, MY); Ahmed Merzouk (Richmond, CA); Abdualrahman Abdualkader (Pahang, MY); Mohamed Alaama (Pahang, MY)
Assignee: Biopep Solutions, Inc.
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Quick Facts
Patent No.
US 8,790,711
App. No.
13/624,856
Granted
Jul 29, 2014
Kind
B2
Abstract

Methods are provided for isolating and using a whole-saliva leech extract. The methods can include feeding a phagostimulatory agent to a leech; inducing a regurgitation in the leech, the inducing including placing the leech in an environment having a temperature of less than about 0° C.; and, collecting an unrefined, whole saliva in the regurgitation of the cooled leech. The methods can include revitalizing the leech by warming it at a temperature ranging from about 5° C. to about 40° C. Stable, lyophilized, whole-saliva extracts of a leech are also provided, the extract having a stable activity when stored for use at a temperature below about −20° C., the extract maintaining at least 70% of the activity for at least 6 months. The extracts can be used to treat solid tumors, treat liquid tumors, treat diabetes, treat a viral disease, treat a parasitic disease, treat an antibacterial disease, or serve as an anti-oxidant.

Claims (35)

1. A method of treating diabetes, comprising administering an effective amount of a whole, leech saliva extract to a subject having diabetes, wherein the extract has a peptide molecular weight distribution with molecular weights of 3496 Daltons or greater; and the administering results in the reduction of an elevated blood glucose concentration when compared to control subjects not receiving the extract.

2. The method of claim 1 , wherein the extract is produced from a process comprising:

feeding a phagostimulatory agent to a leech;

inducing a regurgitation in the leech, the inducing including placing the leech in an environment having a temperature of less than 0° C. or about 0° C.; and,

collecting an unrefined, whole saliva in the regurgitation of the cooled leech.

3. The method of claim 2 , wherein the collecting includes squeezing the leech to increase the amount of unrefined, whole saliva collected.

4. The method of claim 2 , further comprising revitalizing the leech by warming the leech in a water bath having a temperature ranging from about 5° C. to about 40° C.

5. The method of claim 2 , wherein the method further comprises creating a refined, whole-saliva extract; the creating including removing solid components from the unrefined, whole saliva.

6. The method of claim 2 , wherein the method further comprises lyophilizing separate volumes of the refined, whole saliva extract, the volumes not exceeding about 2 ml each.

7. The method of claim 1 , the leech being Hirudinaria manillensis.

8. The method of claim 1 , wherein the extract is a lyophilized, whole saliva extract of a leech produced from a method comprising:

feeding a phagostimulatory agent to a leech;

inducing regurgitation in the leech, the inducing including placing the leech in an environment having a temperature ranging from about −5° C. to about 15° C.;

collecting an unrefined, whole saliva in the regurgitation of the cooled leech;

removing solid components from the unrefined, whole saliva to create a refined, whole saliva; and,

lyophilizing separate volumes of the refined, whole saliva extract, the volumes not exceeding about 2 ml each.

9. The method of claim 8 , wherein the collecting includes squeezing the leech to increase the amount of unrefined, whole saliva collected.

10. The method of claim 8 , further comprising revitalizing the leech by warming the leech in a water bath having a temperature ranging from about 5° C. to about 40° C.

11. The method of claim 8 , the leech being Hirudinaria manillensis.

12. The method of claim 8 , wherein the collecting of the whole saliva yields a peptide molecular weight distribution that ranges from 4276 Daltons to 44386 Daltons.

13. The method of claim 8 , wherein the collecting of the whole saliva yields a peptide molecular weight distribution that ranges from 6289 Daltons to 14244 Daltons.

14. The method of claim 8 , wherein the collecting of the whole saliva yields a peptide molecular weight distribution that ranges from 10812 Daltons to 88210 Daltons.

15. The method of claim 8 , wherein the collecting of the whole saliva yields a peptide molecular weight distribution that ranges from 3496 Daltons to 88210 Daltons.

16. The method of claim 1 , wherein the diabetes is a Type-1 diabetes.

17. The method of claim 1 , wherein the diabetes is a Type-1.5 diabetes.

18. The method of claim 1 , wherein the diabetes is a Type-2 diabetes.

19. The method of claim 1 , wherein the treating of the diabetes includes inhibiting the onset of the diabetes when compared to control subjects not receiving the extract.

20. A method of treating Type-1 diabetes, comprising administering an effective amount of a whole, leech saliva extract to a subject, wherein the extract has a peptide molecular weight distribution with molecular weights of 3496 Daltons or greater; and the administering results in the reduction of an elevated blood glucose concentration when compared to control subjects not receiving the extract.

21. The method of claim 20 , wherein the extract is produced from a process comprising:

feeding a phagostimulatory agent to a leech;

inducing a regurgitation in the leech, the inducing including placing the leech in an environment having a temperature of less than 0° C. or about 0° C.; and,

collecting an unrefined, whole saliva in the regurgitation of the cooled leech.

22. The method of claim 21 , wherein the collecting includes squeezing the leech to increase the amount of unrefined, whole saliva collected.

23. The method of claim 21 , wherein the method further comprises removing solid components from the unrefined, whole saliva to create a refined, whole saliva; and, lyophilizing separate volumes of the refined, whole saliva extract, the volumes not exceeding about 2 ml each.

24. A method of treating a diabetes, comprising administering an effective amount of a whole, leech saliva extract to a subject, the leech being Hirudinaria manillensis wherein the extract has a peptide molecular weight distribution with molecular weights of 3496 Daltons or greater; and the administering results in the reduction of an elevated blood glucose concentration when compared to control subjects not receiving the extract.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 20, 2013
From: MERZOUK, AHMED; GHAWI, ABBAS; ABDUALKADER, ABDUALRAHMAN; ALAAMA, MOHAMED
To: BIOPEP SOLUTIONS, INC.
Reel/Frame 030655/0882 →
Continuity (2)
Provisional Application 61701735 · Sep 17, 2012
Related Publication 20140079799A1 · Mar 20, 2014