IP Library › Granted Patent US 9,078,856
Granted Patent B2
US 9,078,856 · App. 13/703,765 · Granted Jul 14, 2015

Improving efficacy of cancer therapy

Inventors: Charles K. Thodeti (Copley, OH); Donald E. Ingber (Boston, MA)
Assignee: CHILDREN'S MEDICAL CENTER CORPORATION
A61K38/1709A61K31/00A61K31/22A61K31/221A61K31/336A61K31/365A61K38/177A61K45/06A61N5/10
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Quick Facts
Patent No.
US 9,078,856
App. No.
13/703,765
Granted
Jul 14, 2015
Kind
B2
Abstract

Embodiments of the invention provide a method of improving the efficacy of an anti-cancer therapy and a method of treatment of cancer by normalizing angiogenesis in cancer. By enhancing the cell signaling pathway via a TRPV4 receptor in tumor endothelial cells, either by a TRPV4 agonist or by increasing the expression of TRPV4 in the tumor endothelial cells, the tumor endothelial cells behave normally and form normal angiogenic network for better anti-cancer therapy to the tumors.

Claims (6)

1. A method for increasing the efficacy of an anti-cancer treatment in a patient in need thereof, the method comprising administering a TRPV4 agonist or a vector comprising a DNA sequence encoding a human TRVP4 to the patient concurrently with a cancer treatment or subsequently administering the cancer treatment to the patient, wherein the TRPV4 agonist is selected from a group consisting of GSK1016790A, Bisandrographolide A (BAA), RN 1747, AB1644034, α-phorbol 12,13-didecanoate (4αPDD) 5,6-EET, acetylcholine and App441-1.

2. A method for cancer treatment in a patient in need thereof, the method comprising administering a TRPV4 agonist or a vector comprising a DNA sequence encoding a human TRVP4 to the patient concurrently with a cancer treatment or subsequently administering the cancer treatment to the patient, wherein the TRPV4 agonist is selected from a group consisting of GSK1016790A, Bisandrographolide A (BAA), RN 1747, AB1644034, α-phorbol 12,13-didecanoate (4αPDD) 5,6-EET, acetylcholine and App441-1.

3. The method of claim 1 , wherein the cancer treatment is chemotherapy, radiation therapy or immunotherapy.

4. The method of claim 1 , wherein the DNA sequence encoding the human TRVP4 is SEQ. ID. NO. 3, 4 or 5.

5. The method of claim 2 , wherein the cancer treatment is chemotherapy, radiation therapy or immunotherapy.

6. The method of claim 2 , wherein the DNA sequence encoding the human TRVP4 is SEQ. ID. NO. 3, 4 or 5.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 30, 2013
From: INGBER, DONALD E.
To: CHILDREN'S MEDICAL CENTER CORPORATION
Reel/Frame 030906/0259 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 25, 2013
From: THODETI, CHARLES K.
To: NORTHEAST OHIO MEDICAL UNIVERSITY
Reel/Frame 029864/0621 →
Continuity (2)
Provisional Application 61357123 · Jun 22, 2010
Related Publication 20130150432A1 · Jun 13, 2013