IP Library Granted Patent US 9,139,633
Granted Patent B2
US 9,139,633 · App. 13/383,962 · Granted Sep 22, 2015

Mesenchymal stem cell differentiation

Inventors: Kristen Johnson (San Diego, CA); Lori Jennings (San Diego, CA); Peter Schultz (La Jolla, CA)
Assignees: Novartis AG; The Scripps Research Institute
C07K14/515A61K31/728A61K47/48215A61K38/00
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,139,633
App. No.
13/383,962
Granted
Sep 22, 2015
Kind
B2
Abstract

The present invention provides for methods and compositions for treating or preventing arthritis and joint injury.

Claims (23)

1. A method of ameliorating or treating arthritis or joint injury in a mammal, the method comprising administering to a joint of the mammal a composition comprising an effective amount of a C-terminal fibrinogen like domain (FLD) ANGPTL3 polypeptide consisting of:

i. an amino acid sequence at least 95% identical to any one of SEQ ID NO: 5, SEQ ID NO: 6, or SEQ ID NO: 7, or

ii. an amino acid sequence at least 95% identical to any one of SEQ ID NO: 5, SEQ ID NO: 6, or SEQ ID NO: 7 fused to a human serum albumin (HSA), an immunoglobulin heavy chain constant region (Fc), a polyhistidine, a glutathione S transferase (GST), a thioredoxin, a protein A, a protein G, or a maltose binding protein (MBP);

thereby ameliorating or treating arthritis or joint injury in the mammal.

2. The method of claim 1 , wherein the polypeptide is PEGylated.

3. The method of claim 1 , wherein the individual has arthritis or joint injury.

4. The method of claim 1 , wherein the arthritis is selected from the group consisting of osteoarthritis, trauma arthritis, and autoimmune arthritis.

5. The method of claim 1 , wherein the mammal is a human, a dog, or a cat.

6. The method of claim 1 , wherein the composition further comprises hyaluronic acid.

7. The method of claim 1 , wherein the amino acid sequence comprises SEQ ID NO: 5, 6 or 7.

8. The method of claim 1 , wherein the amino acid sequence is SEQ ID NO: 5, SEQ ID NO: 6, or SEQ ID NO: 7.

9. A method of inducing differentiation of mesenchymal stem cells into chondrocytes, the method comprising contacting mesenchymal stem cells with a sufficient amount of a C-terminal fibrinogen like domain (FLD) ANGPTL3 polypeptide consisting of:

i. an amino acid sequence at least 95% identical to any one of SEQ ID NO: 5, SEQ ID NO: 6, or SEQ ID NO: 7, or

ii. an amino acid sequence at least 95% identical to any one of SEQ ID NO: 5, SEQ ID NO: 6, or SEQ ID NO: 7 fused to a human serum albumin (HSA), an immunoglobulin heavy chain constant region (Fc), a polyhistidine, a glutathione S transferase (GST), a thioredoxin, a protein A, a protein G, or a maltose binding protein (MBP);

to induce differentiation of the stem cells into chondrocytes.

10. The method of claim 9 , wherein the polypeptide is PEGylated.

11. The method of claim 9 , wherein the method is performed in vitro.

12. The method of claim 9 , wherein the method is performed in vivo and the stem cells are present in a mammal.

13. The method of claim 12 , wherein the mammal is a human, a dog, or a cat.

14. The method of claim 12 , wherein the mammal has arthritis or joint injury.

15. The method of claim 14 , wherein the arthritis is selected from the group consisting of osteoarthritis, trauma arthritis, and autoimmune arthritis.

16. The method of claim 9 wherein the amino acid sequence comprises SEQ ID NO: 5, SEQ ID NO: 6 or SEQ ID NO: 7.

17. The method of claim 9 , wherein the amino acid sequence is SEQ ID NO: 5, SEQ ID NO: 6, or SEQ ID NO: 7.

Assignments (4)
MERGER Recorded Apr 22, 2015
From: IRM LLC
To: NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD.
Reel/Frame 035468/0184 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 22, 2015
From: NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD.
To: NOVARTIS AG
Reel/Frame 035468/0264 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 2, 2012
From: NOVARTIS INSTITUTE FOR FUNCTIONAL GENOMICS, INC., DBA GENOMICS INSTITUTE OF THE NOVARTIS RESEARCH FOUNDATION
To: IRM LLC
Reel/Frame 028476/0433 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 21, 2012
From: JENNINGS, LORI; JOHNSON, KRISTEN
To: NOVARTIS INSTITUTE FOR FUNCTIONAL GENOMICS, INC., DBA GENOMICS INSTITUTE OF THE NOVARTIS RESEARCH FOUNDATION
Reel/Frame 028421/0638 →
Continuity (2)
Provisional Application 61225293 · Jul 14, 2009
Related Publication 20120177644A1 · Jul 12, 2012