IP Library Granted Patent US 9,683,000
Granted Patent B2
US 9,683,000 · App. 15/017,329 · Granted Jun 20, 2017

Carbonate prodrugs and methods of using the same

Inventors: Naweed Muhammad (Fremont, CA); Keith R. Bley (Menlo Park, CA)
Assignee: Acorda Therapeutics, Inc.
C07F9/096A61K31/661A61K47/48084C07C233/25C07F9/11
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Quick Facts
Patent No.
US 9,683,000
App. No.
15/017,329
Granted
Jun 20, 2017
Kind
B2
Abstract

The present invention provides carbonate prodrugs which comprise a carbonic phosphoric anhydride prodrug moiety attached to the hydroxyl or carboxyl group of a parent drug moiety. The prodrugs may provide improved physicochemical properties over the parent drug. Also provided are methods of treating a disease or condition that is responsive to the parent drug using the carbonate prodrugs, as well as kits and unit dosages.

Claims (2)

1. A compound of the formula

or a salt thereof.

Assignments (4)
RELEASE OF SECURITY INTEREST Recorded May 31, 2017
From: JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT
To: NEURONEX, INC.; CIVITAS THERAPEUTICS, INC.; ACORDA THERAPEUTICS, INC.
Reel/Frame 042643/0878 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 12, 2017
From: MUHAMMAD, NAWEED; BLEY, KEITH R.
To: NEUROGESX, INC.
Reel/Frame 040973/0563 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 12, 2017
From: NEUROGESX, INC.
To: ACORDA THERAPEUTICS, INC.
Reel/Frame 041355/0080 →
SECURITY INTEREST Recorded Jun 10, 2016
From: ACORDA THERAPEUTICS, INC.; CIVITAS THERAPEUTICS, INC.; NEURONEX, INC.
To: JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT
Reel/Frame 038950/0436 →
Continuity (5)
Continuation 14629324 · Feb 23, 2015
Continuation 14252683 · Apr 14, 2014
Division 12993089
Provisional Application 61054765 · May 20, 2008
Related Publication 20170008916A1 · Jan 12, 2017