IP Library › Granted Patent US 9,925,186
Granted Patent B2
US 9,925,186 · App. 14/814,018 · Granted Mar 27, 2018

Method of treating metabolic disorders and depression with dopamine receptor agonists

Inventor: Anthony H. Cincotta (Tiverton, RI)
Assignee: VeroScience LLC
A61K31/4985A61K31/00A61K31/48A61K45/06
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Quick Facts
Patent No.
US 9,925,186
App. No.
14/814,018
Granted
Mar 27, 2018
Kind
B2
Abstract

This invention relates to methods and formulations for treating metabolic disorders and depression. In some embodiments, the methods comprise administering a dopamine receptor agonist and an anti-depressant.

Claims (15)

1. The method of treating a patient afflicted with type 2 diabetes and depression that is taking a serotonin enhancing anti-depressant comprising administering to a patient in need of such treatment a therapeutically effective amount of one or more dopamine receptor agonists daily at a first pre-determined time of day in the morning.

2. The method of claim 1 , wherein the pre-determined time of day is between 0400 and 1200 hoursin the morning.

3. The method of claim 2 , wherein the pre-determined time of day is upon waking.

4. The method of claim 1 , wherein the dopamine receptor agonist is at least one of a dopamine D1 receptor agonist or a dopamine D2 receptor agonist.

5. The method of claim 1 , wherein the dopamine receptor agonist is an ergot-related compound.

6. The method of claim 1 wherein the dopamine receptor agonist is selected from the group consisting of lisuride, terguride, dihydroergotoxine (hydergine), and bromocriptine.

7. The method of claim 1 wherein the dopamine receptor agonist is bromocriptine.

8. The method of claim 4 wherein the dopamine receptor agonist is a dopamine D1 receptor agonist.

9. The method of claim 4 wherein the dopamine receptor agonist is a dopamine D2 receptor agonist.

10. The method of claim 8 wherein the therapeutically effective amount is between about 0.01 to about 50.0 mg/kg.

11. The method of claim 10 wherein the therapeutically effective amount is between about 0.1 to about 25.0 mg/kg.

12. The method of treating a patient afflicted with type-2 diabetes and depression that is taking a serotonin enhancing anti-depressant comprising administering to a patient in need of such treatment a therapeutically effective amount of a D1 dopamine receptor agonist and a D2 dopamine receptor agonist once daily at a predetermined time for bioavailability in the morning and at a point after the peak in plasma prolactin level.

13. A method of treating a patient suffering from pre-diabetes and depression that is taking a serotonin enhancing anti-depressant comprising administering to a patient in need of such treatment a therapeutically effective amount of one or more dopamine receptor agonists daily at a first pre-determined time of day in the morning.

14. The method of claim 13 wherein the pre-determined time of day is between 0400 and 1200 hours in the morning.

15. The method of claim 13 wherein the predetermined time of day is within 2 hours of waking.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 9, 2018
From: CINCOTTA, ANTHONY H.
To: VEROSCIENCE LLC
Reel/Frame 044886/0505 →
Continuity (4)
Division 13774739 · Feb 22, 2013
Continuation 12144617 · Jun 23, 2008
Provisional Application 60945555 · Jun 21, 2007
Related Publication 20150335641A1 · Nov 26, 2015