IP Library Granted Patent US 9,125,875
Granted Patent B2
US 9,125,875 · App. 14/567,267 · Granted Sep 8, 2015

Use of the cathelicidin LL-37 and derivatives thereof for wound healing

Inventors: Mona Ståhle-Bäckdahl (Stockholm, SE); Johan Heilborn (Stockholm, SE); Anders Carlsson (Stockholm, SE); Conny Bogentoft (Hasselby, SE)
Assignee: Lipopeptide AB
A61K38/1709A61K9/1272A61K38/16C07K14/47C07K14/4723C12N5/0018C12N5/0629C12N2500/32C12N2500/36Y10S514/938
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,125,875
App. No.
14/567,267
Granted
Sep 8, 2015
Kind
B2
Abstract

Use of the antimicrobial cathelicidin peptide II-37, N-terminal fragments of LL-37 or extended sequences of LL-37 having 1-3 amino acids in the C-terminal end, for stimulating proliferation of epithelial and stromal cells and thereby healing of wounds, such as chronic ulcers. The cytotoxic effect of LL-37 may be reduced by including a bilayer-forming polar lipid, especially a digalactosyldiacylglycerol, in pharmaceutical compositions and growth media comprising LL-37.

Claims (9)

1. A method for stimulating proliferation of epithelial cells in a chronic ulcer due to diabetes, comprising administering an effective amount of a peptide LL-37 (SEQ ID NO: 1) or a pharmaceutically acceptable salt thereof to a subject in need of such treatment.

2. The method according to claim 1 , wherein said peptide LL-37 (SEQ ID NO: 1) is in the form of the acetate salt.

3. The method of claim 1 wherein the peptide LL-37 (SEQ ID NO: 1) is administered topically to the chronic ulcer.

4. A method for stimulating epithelial regeneration in a chronic ulcer due to diabetes, comprising administering an effective amount of a peptide LL-37 (SEQ ID NO: 1) or a pharmaceutically acceptable salt thereof to a subject in need of such treatment.

5. The method according to claim 4 , wherein said peptide LL-37 (SEQ ID NO: 1) is in the form of the acetate salt.

6. The method of claim 4 wherein the peptide LL-37 (SEQ ID NO: 1) is administered topically to the chronic ulcer.

7. A method for stimulating re-epithelialization in a chronic ulcer due to diabetes, comprising administering an effective amount of a peptide LL-37 (SEQ ID NO: 1) or a pharmaceutically acceptable salt thereof to a subject in need of such treatment.

8. The method according to claim 7 , wherein said peptide LL-37 (SEQ ID NO: 1) is in the form of the acetate salt.

9. The method of claim 7 wherein the peptide LL-37 (SEQ ID NO: 1) is administered topically to the chronic ulcer.

Assignments (2)
CHANGE OF NAME Recorded Dec 10, 2018
From: LIPOPEPTIDE AB
To: PROMORE PHARMA AB
Reel/Frame 047763/0465 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 3, 2015
From: STAHLE-BACKDAHL, MONA; HEILBORN, JOHAN; CARLSSON, ANDERS; BOGENTOFT, CONNY
To: LIPOPEPTIDE AB
Reel/Frame 036486/0749 →
Priority Claims (1)
SE 0300207 · Jan 29, 2003 · national
Continuity (6)
Continuation 13938120 · Jul 9, 2013
Division 13193131 · Jul 28, 2011
Division 12232215 · Sep 12, 2008
Division 10543659
Provisional Application 60444964 · Feb 5, 2003
Related Publication 20150094256A1 · Apr 2, 2015