IP Library Granted Patent US 9,532,992
Granted Patent B2
US 9,532,992 · App. 14/742,466 · Granted Jan 3, 2017

Substituted benzene compounds

Inventors: Kevin Wayne Kuntz (Woburn, MA); John Emmerson Campbell (Cambridge, MA); Masashi Seki (Tsukuba, JP)
Assignee: Epizyme, Inc.
A61K31/5375A61K31/4412A61K31/4545A61K31/5377C07D213/64C07D401/12C07D405/12C07D405/14
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Quick Facts
Patent No.
US 9,532,992
App. No.
14/742,466
Granted
Jan 3, 2017
Kind
B2
Abstract

The present invention relates to substituted benzene compounds. The present invention also relates to pharmaceutical compositions containing these compounds and methods of treating cancer by administering these compounds and pharmaceutical compositions to subjects in need thereof. The present invention also relates to the use of such compounds for research or other non-therapeutic purposes.

Claims (32)

1. A method comprising administering to a subject in need thereof

or

a pharmaceutically acceptable salt thereof at a dosage ranging from about 0.01 mg/kg per day to about 5000 mg/kg per day.

2. The method of claim 1 , wherein the subject has been diagnosed or identified as having cancer or a precancerous condition.

3. The method of claim 2 , wherein the cancer is lymphoma, malignant rhabdoid tumor, a hematological cancer, leukemia, or melanoma.

4. The method of claim 3 , wherein the lymphoma is selected from diffuse large B-cell lymphoma (DLBCL), non-Hodgkin's lymphoma (NHL), and follicular lymphoma.

5. The method of claim 2 , wherein the cancer is malignant rhabdoid tumor.

6. The method of claim 1 , wherein the compound is

or a pharmaceutically acceptable salt thereof.

7. The method of claim 1 , wherein the subject is human or non-human mammal.

8. The method of claim 7 , wherein the non-human mammal is a primate, dog, cow, or pig.

9. The method of claim 1 , wherein the subject is a dog.

10. A method comprising administering to a subject in need thereof

or

a pharmaceutically acceptable salt thereof at a dosage ranging from about 0.01 mg/kg per day to about 5000 mg/kg per day.

11. The method of claim 10 , wherein the subject has been diagnosed or identified as having cancer or a precancerous condition.

12. The method of claim 11 , wherein the cancer is lymphoma, malignant rhabdoid tumor, a hematological cancer, leukemia, or melanoma.

13. The method of claim 12 , wherein the lymphoma is selected from diffuse large B-cell lymphoma (DLBCL), non-Hodgkin's lymphoma (NHL), and follicular lymphoma.

14. The method of claim 11 , wherein the cancer is malignant rhabdoid tumor.

15. The method of claim 10 , wherein the subject is human or non-human mammal.

16. The method of claim 15 , wherein the non-human mammal is a primate, dog, cow, or pig.

17. The method of claim 10 , wherein the subject is a dog.

18. A method comprising administering to a subject in need thereof

or

a pharmaceutically acceptable salt thereof at a dosage ranging from about 0.01 mg/kg per day to about 5000 mg/kg per day.

19. The method of claim 18 , wherein the subject has been previously diagnosed or identified as having cancer or a precancerous condition.

20. The method of claim 19 , wherein the cancer is lymphoma, malignant rhabdoid tumor, a hematological cancer, leukemia, or melanoma.

21. The method of claim 20 , wherein the lymphoma is selected from diffuse large B-cell lymphoma (DLBCL), non-Hodgkin's lymphoma (NHL), and follicular lymphoma.

22. The method of claim 18 , wherein the cancer is malignant rhabdoid tumor.

23. The method of claim 18 , wherein the subject is human or non-human mammal.

24. The method of claim 23 , wherein the non-human mammal is a primate, dog, cow, or pig.

25. The method of claim 18 , wherein the subject is a dog.

Assignments (5)
TERMINATION AND RELEASE OF SECURITY INTEREST IN PATENTS AT REEL/FRAME: 051057/0848 Recorded Aug 13, 2022
From: BIOPHARMA CREDIT PLC
To: EPIZYME, INC.
Reel/Frame 061165/0501 →
SECURITY INTEREST Recorded Nov 19, 2019
From: EPIZYME, INC.
To: BIOPHARMA CREDIT PLC
Reel/Frame 051057/0848 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 30, 2015
From: EISAI R&D MANAGEMENT CO., LTD.
To: EPIZYME, INC.
Reel/Frame 035939/0677 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 24, 2015
From: KUNTZ, KEVIN WAYNE; CAMPBELL, JOHN EMMERSON
To: EPIZYME, INC.
Reel/Frame 035898/0685 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 24, 2015
From: SEKI, MASASHI
To: EISAI R&D MANAGEMENT CO., LTD.
Reel/Frame 035898/0723 →
Continuity (7)
Continuation 14639878 · Mar 5, 2015
Continuation 14054695 · Oct 15, 2013
Provisional Application 61714140 · Oct 15, 2012
Provisional Application 61714145 · Oct 15, 2012
Provisional Application 61780703 · Mar 13, 2013
Provisional Application 61786277 · Mar 14, 2013
Related Publication 20150352119A1 · Dec 10, 2015