IP Library Granted Patent US 9,844,219
Granted Patent B2
US 9,844,219 · App. 15/223,748 · Granted Dec 19, 2017

Alpha-keto peracids and methods for producing and using the same

Inventors: Edwin D. Neas (Nunn, CO); John D. Skinner (Fort Collins, CO)
Assignee: CHD BIOSCIENCE, INC.
A01N37/42A61K31/13A61K31/327A61K33/40A61K45/06C07C407/00C07C409/24C07C2601/08
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Quick Facts
Patent No.
US 9,844,219
App. No.
15/223,748
Granted
Dec 19, 2017
Kind
B2
Abstract

The present invention provides α-keto peracids and methods for producing and using the same. In particular, α-keto peracids are useful as antimicrobial agents.

Claims (24)

1. An antimicrobial composition comprising the products of a method comprising contacting an α-keto carboxylic acid or a salt thereof with an oxidizing agent to form a mixture, and allowing the mixture to stand at a temperature of −30° C. to 4° C., wherein the products comprise an α-keto peracid.

2. The antimicrobial composition of claim 1 , wherein the temperature is −10° C. to 4° C.

3. The antimicrobial composition of claim 1 , wherein the oxidizing agent is at a concentration of 1M to 12M.

4. The antimicrobial composition of claim 1 , wherein the oxidizing agent is at a concentration of 1M to 7M.

5. The antimicrobial composition of claim 1 , wherein the mixture is allowed to stand for a reaction time of 4 hours to 12 hours.

6. The antimicrobial composition of claim 1 , wherein the mixture is allowed to stand for a reaction time of 10 hours to 12 hours.

7. The antimicrobial composition of claim 1 , wherein the oxidizing agent is selected from the group consisting of hydrogen peroxide, barium peroxide, sodium carbonate peroxide, calcium peroxide, sodium perborate, lithium peroxide, magnesium peroxide strontium peroxide, zinc peroxide, and potassium superoxide.

8. The antimicrobial composition of claim 1 , wherein the ratio of oxidizing agent to α-keto carboxylic acid is 0.5:1 to 6:1.

9. The antimicrobial composition of claim 1 , wherein the ratio of oxidizing agent to α-keto carboxylic acid is 0.5 to 2:1.

10. The antimicrobial composition of claim 1 , wherein the ratio of oxidizing agent to α-keto carboxylic acid is 2:1 to 6:1.

11. The antimicrobial composition of claim 1 further comprising at least one of water and one or more additional antimicrobial agent selected from organic acids, peroxides, alcohols, ethers, hydrogen peroxide, dichloracetic acid, diacetone alcohol, and butylene glycol monomethyl ether.

12. The antimicrobial composition of claim 1 , wherein the α-keto carboxylic acid or a salt thereof is selected from the group consisting of pyruvic acid, α-ketobutanoic acid, and α-ketovaleric acid, or a salt thereof, the oxidizer is hydrogen peroxide, the temperature is between −30° C. and 10° C., and the mixture is allowed to stand until all α-keto carboxylic acid is dissolved into solution.

13. The antimicrobial composition of claim 12 , wherein the α-keto carboxylic acid or a salt thereof is pyruvic acid or a salt thereof.

14. The antimicrobial composition of claim 1 , wherein:

the temperature is −10° C. to 4° C.;

the oxidizing agent is at a concentration of 1M to 12M;

the mixture is allowed to stand for a reaction time of 4 hours to 12 hours; and

the ratio of oxidizing agent to α-keto carboxylic acid is 0.5:1 to 6:1.

15. The antimicrobial composition of claim 14 , wherein the oxidizing agent is selected from the group consisting of hydrogen peroxide, barium peroxide, sodium carbonate peroxide, calcium peroxide, sodium perborate, lithium peroxide, magnesium peroxide strontium peroxide, zinc peroxide, and potassium superoxide.

16. The antimicrobial composition of claim 15 , wherein the oxidizing agent is hydrogen peroxide.

17. The antimicrobial composition of claim 16 , wherein the products comprise an α-keto alkylperacid of the formula: HOO—C(═O)—C(═O)—R or a salt thereof, where R is alkyl of at least one carbon atom.

18. The antimicrobial composition of claim 17 , wherein R is selected from the group consisting of ethyl, isopropyl, propyl, butyl, isobutyl, sec-butyl, pentyl, isopentyl, neopentyl, and n-hexyl.

19. The antimicrobial composition of claim 16 , wherein the oxidizing agent is at a concentration of 1M to 7M, and reaction time is 10 hours to 12 hours.

20. The antimicrobial composition of claim 19 , wherein the α-keto carboxylic acid is selected from the group consisting of α-keto pyruvic acid, α-keto butyric acid, and α-keto valeric acid.

Assignments (3)
CHANGE OF NAME Recorded Jan 31, 2022
From: CHD BIOSCIENCE, INC.
To: ARMIS BIOPHARMA, INC.
Reel/Frame 058834/0571 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 1, 2016
From: NEAS, EDWIN D.; SKINNER, JOHN D.
To: CHATA BIOSYSTEMS, INC.
Reel/Frame 039616/0350 →
CHANGE OF NAME Recorded Sep 1, 2016
From: CHATA BIOSYSTEMS, INC.
To: CHD BIOSCIENCE, INC.
Reel/Frame 039900/0598 →
Continuity (8)
Continuation 14671223 · Mar 27, 2015
Continuation 13860680 · Apr 11, 2013
Continuation 12618605 · Nov 13, 2009
Continuation 13898126 · May 20, 2013
Continuation 12760940 · Apr 15, 2010
Continuation In Part 12618605 · Nov 13, 2009
Provisional Application 61199944 · Nov 20, 2008
Related Publication 20160330958A1 · Nov 17, 2016