IP Library Granted Patent US 10,688,122
Granted Patent B2
US 10,688,122 · App. 15/279,301 · Granted Jun 23, 2020

Thiol and disulfide-containing agents for increasing meibomian gland lipid secretion

Inventors: Shimon Amselem (Rehovot, IL); Yair Alster (Tel Aviv, IL); Doron Friedman (Carme-Yosef, IL); Omer Rafaeli (Udim, IL)
Assignee: AZURA OPHTHALMICS LTD.
A61K33/04A61K9/0048A61K31/095A61K31/19A61K31/198A61K31/20A61K31/325A61K31/401A61K31/575A61K31/683A61K45/06A61K47/06A61K47/44
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Quick Facts
Patent No.
US 10,688,122
App. No.
15/279,301
Granted
Jun 23, 2020
Kind
B2
Abstract

Described herein are compositions and methods for the increasing the quantity of lipids secreted from meibomian glands. Such compositions and methods are useful for the treatment of meibomian gland dysfunction and disorders resulting therefrom.

Claims (11)

1. A method for increasing lipid secretion from a meibomian gland, comprising topically administering to the eyelid margin of the patient in need thereof an ophthalmic composition comprising an ophthalmically-acceptable carrier and an effective amount of at least one agent which increases lipogenesis in the meibomian gland or increases lipid secretion from the meibomian gland, wherein the agent is captopril or selenocysteine.

2. The method of claim 1 , wherein the ophthalmically-acceptable carrier comprises at least one ophthalmically-acceptable excipient.

3. The method of claim 1 , further comprising the step of administering to the patient a keratolytic agent.

4. The method of claim 3 , wherein the keratolytic agent is selected from the group consisting of benzoyl peroxide, coal tar, dithranol, salicylic acid, selenium disulfide, alpha-hydroxy acid, urea, boric acid, retinoic acid, lactic acid, sodium thioglycolate or allantoin.

5. A method for increasing lipid secretion from a meibomian gland, comprising topically administering to the eyelid margin of the patient in need thereof an ophthalmic composition comprising an effective amount of a single agent which increases lipogenesis in the meibomian gland or increases lipid secretion from the meibomian gland, wherein the agent is captopril or selenocysteine.

6. The method of claim 5 , further comprising the step of administering to the patient a keratolytic agent.

7. The method of claim 6 , wherein the keratolytic agent is selected from the group consisting of benzoyl peroxide, coal tar, dithranol, salicylic acid, selenium disulfide, alpha-hydroxy acid, urea, boric acid, retinoic acid, lactic acid, sodium thioglycolate or allantoin.

8. The method of claim 1 , wherein the agent is captopril.

9. The method of claim 1 , wherein the agent is selenocysteine.

10. The method of claim 5 , wherein the agent is captopril.

11. The method of claim 5 , wherein the agent is selenocysteine.

Assignments (2)
CHANGE OF NAME Recorded Jan 16, 2020
From: M.G. THERAPEUTICS LTD.
To: AZURA OPHTHALMICS LTD.
Reel/Frame 051625/0912 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 8, 2016
From: ALSTER, YAIR; AMSELEM, SHIMON; FRIEDMAN, DORON; RAFAELI, OMER
To: M.G. THERAPEUTICS LTD.
Reel/Frame 040259/0077 →
Continuity (3)
Provisional Application 62233941 · Sep 28, 2015
Provisional Application 62233906 · Sep 28, 2015
Related Publication 20170087179A1 · Mar 30, 2017
Cited By (9)
US 12,213,964 US 12,257,263 US 12,364,685 US 12,427,158 US 12,447,162 US 12,458,661 US 12,502,377 US 12,661,339 US 12,697,352