IP Library Granted Patent US 10,335,426
Granted Patent B2
US 10,335,426 · App. 15/702,529 · Granted Jul 2, 2019

N-acetyl mannosammine as a therapeutic agent

Inventors: Marjan Huizing (Santa Cruz, CA); William A. Gahl (Kensington, MD); Irini Manoli (Rockville, MD); Enriko Klootwijk (London, GB)
Assignee: THE UNITED STATES OF AMERICA, as represented by the Secretary, Department of Health and Human Services
A61K31/7008A61K31/7012
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Quick Facts
Patent No.
US 10,335,426
App. No.
15/702,529
Granted
Jul 2, 2019
Kind
B2
Abstract

The invention relates to compositions and methods for treating kidney and muscle dysfunction that involves use of therapeutic amounts of N-acetyl mannosamine.

Claims (10)

1. A method of treating a condition or disease in a mammal in need thereof comprising selecting a subject with the condition or disease, and administering to the subject an effective amount of N-acetyl mannosamine or a derivative thereof, to the mammal, wherein the derivative consists of Formula I.

wherein R 1 , R 3 , R 4 , or R 5 is hydrogen, lower alkanoyl, carboxylate or lower alkyl; R 2 is lower alkyl, lower alkanoylalkyl, lower alkyl alkanoyloxy; and the condition or disease is diabetic nephropathy.

2. The method of claim 1 , comprising administering a therapeutic amount of N-acetyl mannosamine to the mammal.

3. The method of claim 2 , wherein the therapeutic amount is about 0.1 g to about 50 g N-acetyl mannosamine per day.

4. The method of claim 2 , wherein the therapeutic amount is administered in a unit dosage of about 0.01 g to about 50 g N-acetyl mannosamine per unit dosage.

5. The method of claim 1 , comprising sustained release of the sialic acid precursor, N-acetyl mannosamine or a derivative thereof.

6. The method of claim 1 , comprising topical administration of the sialic acid precursor, N-acetyl mannosamine or a derivative thereof.

7. The method of claims 2 , wherein the N-acetyl mannosamine is administered orally to the mammal.

8. The method of claim 2 , wherein the N-acetyl mannosamine is microencapsulated.

9. The method of claim 2 , wherein the method decreases proteinuria in the mammal.

Assignments (3)
CHANGE OF NAME Recorded Apr 19, 2019
From: GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES
To: THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES
Reel/Frame 048941/0906 →
CHANGE OF NAME Recorded Apr 8, 2019
From: GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES
To: THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES
Reel/Frame 048824/0246 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 20, 2019
From: HUIZING, MARJAN; GAHL, WILLIAM A.; MANOLI, IRINI; KLOOTWIJK, ENRIKO
To: GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICE
Reel/Frame 048383/0802 →
Continuity (5)
Continuation 14754304 · Jun 29, 2015
Continuation 13791576 · Mar 8, 2013
Continuation 12530433
Provisional Application 60932451 · May 31, 2007
Related Publication 20180117072A1 · May 3, 2018