IP Library Granted Patent US 10,858,323
Granted Patent B2
US 10,858,323 · App. 16/026,651 · Granted Dec 8, 2020

HDAC inhibitors for the treatment of diabetic peripheral neuropathy

Inventors: Olga Golonzhka (Watertown, MA); Matthew B. Jarpe (Quincy, MA)
Assignee: REGENACY PHARMACEUTICALS, LLC
C07D239/42A61K31/164A61K31/337A61K31/495A61K31/505
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Quick Facts
Patent No.
US 10,858,323
App. No.
16/026,651
Granted
Dec 8, 2020
Kind
B2
Abstract

The invention relates to HDAC inhibitors for use in the treatment of diabetic peripheral neuropathy in a subject in need thereof. Also provided herein are methods for treating diabetic peripheral neuropathy in a subject in need thereof comprising administering to the subject a therapeutically effective amount of an HDAC inhibitor.

Claims (9)

1. A method for treating diabetic peripheral neuropathy in a subject in need thereof comprising administering to the subject a therapeutically effective amount of an HDAC6-specific inhibitor.

2. The method of claim 1 , wherein the HDAC6-specific inhibitor is a compound of Formula II:

or a pharmaceutically acceptable salt thereof,

wherein ring B is aryl or heteroaryl optionally substituted by OH, halo, or C 1-6 -alkyl;

R 1 is aryl or heteroaryl optionally substituted by OH, halo, or C 1-6 -alkyl; and

R is H or C 1-6 -alkyl.

3. The method of claim 2 , wherein the compound of Formula II is:

or a pharmaceutically acceptable salt thereof.

4. The method of claim 1 , wherein the HDAC6-specific inhibitor is administered by oral administration.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 25, 2020
From: GOLONZHKA, OLGA; JARPE, MATTHEW B.
To: ACETYLON PHARMACEUTICALS, INC.
Reel/Frame 052221/0880 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 25, 2020
From: ACETYLON PHARMACEUTICALS, INC.
To: REGENACY PHARMACEUTICALS, LLC
Reel/Frame 052222/0226 →
Continuity (4)
Continuation 15335971 · Oct 27, 2016
Provisional Application 62246965 · Oct 27, 2015
Provisional Application 62281990 · Jan 22, 2016
Related Publication 20190106392A1 · Apr 11, 2019
Cited By (2)
US 12,201,617 US 12,312,345