IP Library Granted Patent US 10,696,679
Granted Patent B2
US 10,696,679 · App. 16/042,085 · Granted Jun 30, 2020

Methods and compounds for treating paramyxoviridae virus infections

Inventors: Richard L. Mackman (Millbrae, CA); Jay P. Parrish (Redwood City, CA); Adrian S. Ray (Redwood City, CA); Dorothy Agnes Theodore (Castro Valley, CA)
Assignee: GILEAD SCIENCES, INC.
C07D487/04A61K9/0078A61K31/706A61K45/06C07F9/6561C07H7/06C07H19/04
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Quick Facts
Patent No.
US 10,696,679
App. No.
16/042,085
Granted
Jun 30, 2020
Kind
B2
Abstract

Provided are methods for treating Paramyxoviridae virus infections by administering ribosides, riboside phosphates and prodrugs thereof, of Formula I: wherein the 1′ position of the nucleoside sugar is substituted. The compounds, compositions, and methods provided are particularly useful for the treatment of Human parainfluenza and Human respiratory syncytial virus infections.

Claims (10)

1. A method of treating a Paramyxoviridae infection, comprising administering to a human subject in need thereof a therapeutically effective amount of a compound of Formula

or a pharmaceutically acceptable salt or ester, thereof.

2. The method of claim 1 further comprising administering a therapeutically effective amount of at least one other therapeutic agent or composition thereof selected from the group consisting of a corticosteroid, an anti-inflammatory signal transduction modulator, a β2-adrenoreceptor agonist bronchodilator, an anticholinergic, a mucolytic agent, hypertonic saline and other drugs for treating Paramyxoviridae virus infections; or mixtures thereof.

3. The method of claim 2 wherein the at least one other therapeutic agent is ribavirin, palivizumab, motavizumab, RSV-IGIV, MEDI-557, A-60444, MDT-637 or BMS-433771 or mixtures thereof.

4. The method of claim 1 wherein the Paramyxoviridae infection is caused by a type 1 or 3 Human parainfluenza virus.

5. The method of claim 1 wherein the Paramyxoviridae infection is caused by a Pneumovirinae virus.

6. The method of claim 1 wherein the Paramyxoviridae infection is caused by a Human respiratory syncytial virus.

7. The method of claim 1 comprising administering the compound of Formula

or a pharmaceutically acceptable salt thereof.

8. The method of claim 1 comprising administering the compound of Formula

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 1, 2018
From: MACKMAN, RICHARD L.; PARRISH, JAY P.; RAY, ADRIAN S.; THEODORE, DOROTHY AGNES
To: GILEAD SCIENCES, INC.
Reel/Frame 046527/0849 →
Continuity (4)
Division 14613719 · Feb 4, 2015
Continuation 13189373 · Jul 22, 2011
Provisional Application 61366609 · Jul 22, 2010
Related Publication 20190055251A1 · Feb 21, 2019
Cited By (6)
US 12,297,226 US 12,357,577 US 12,404,289 US 12,448,383 US 12,509,466 US 12,655,172