IP Library Granted Patent US 10,940,110
Granted Patent B2
US 10,940,110 · App. 16/217,765 · Granted Mar 9, 2021

Method and system for the treatment of chronic COPD with nebulized anticholinergic administrations

Inventors: William Gerhart (La Mesa, CA); Ahmet Tutuncu (San Diego, CA)
Assignee: SUNOVION RESPIRATORY DEVELOPMENT INC.
A61K9/0078A61K31/00A61K31/40A61K31/4015A61K31/56A61M11/00
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Quick Facts
Patent No.
US 10,940,110
App. No.
16/217,765
Granted
Mar 9, 2021
Kind
B2
Abstract

A method is provided for improving lung function in COPD by administering a muscarinic antagonist with a high efficiency nebulizer.

Claims (18)

1. A pharmaceutical composition, comprising an aqueous solution of glycopyrrolate having a volume of about 0.7 mL to about 1.0 mL, a glycopyrrolate concentration of about 25 μg/mL to about 400 μg/mL, and a pH of about 3 to about 5, wherein the solution is free of other bronchodilating agents and is substantially free of preservatives.

2. The pharmaceutical composition of claim 1 , further comprising an organic acid.

3. The pharmaceutical composition of claim 2 , wherein the organic acid is citric acid or a pharmaceutically acceptable salt thereof.

4. The pharmaceutical composition of claim 1 , wherein the solution is substantially free of benzyl alcohol.

5. The pharmaceutical composition of claim 1 , wherein the glycopyrrolate concentration is about 25 μg/mL.

6. The pharmaceutical composition of claim 1 , wherein the volume is about 1 mL.

7. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition is contained in a single dose ampule.

8. The pharmaceutical composition of claim 1 , comprising an aqueous solution of glycopyrrolate having a volume of about 1.0 mL, a glycopyrrolate concentration of about 25 μg/mL, and a pH of about 3 to about 5, wherein the solution is free of other bronchodilating agents and is substantially free of preservatives.

9. The pharmaceutical composition of claim 8 , wherein said aqueous solution further comprises citric acid or a pharmaceutically acceptable salt thereof.

10. A method of treating chronic obstructive pulmonary disease (COPD) in a subject comprising administering to the subject a pharmaceutical composition via a high efficiency nebulizer, wherein the pharmaceutical composition comprises an aqueous solution of glycopyrrolate having a volume of about 0.7 mL to about 1.0 mL, a glycopyrrolate concentration of about 25 μg/mL to about 400 μg/mL, and a pH of about 3 to about 5, wherein the solution is free of other bronchodilating agents and is substantially free of preservatives.

11. The method of claim 10 , wherein the pharmaceutical composition further comprises an organic acid.

12. The method of claim 11 , wherein the organic acid is citric acid or a pharmaceutically acceptable salt thereof.

13. The method of claim 10 , wherein the solution is substantially free of benzyl alcohol.

14. The method of claim 10 , wherein the glycopyrrolate concentration is about 25 μg/mL.

15. The method of claim 10 , wherein the volume is about 1 mL.

16. The method of claim 10 , wherein the pharmaceutical composition is contained in a single dose ampule.

17. The method of claim 10 , wherein the pharmaceutical composition comprises an aqueous solution of glycopyrrolate having a volume of about 1.0 mL, a glycopyrrolate concentration of about 25 μg/mL, and a pH of about 3 to about 5, wherein the solution is free of other bronchodilating agents and is substantially free of preservatives.

18. The method of claim 17 , wherein said aqueous solution further comprises citric acid or a pharmaceutically acceptable salt thereof.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 13, 2018
From: GERHART, WILLIAM; TUTUNCU, AHMET
To: ELEVATION PHARMACEUTICALS, INC.
Reel/Frame 047767/0251 →
MERGER Recorded Dec 13, 2018
From: ELEVATION PHARMACEUTICALS, INC.
To: SUNOVION RESPIRATORY DEVELOPMENT INC.
Reel/Frame 047767/0287 →
Continuity (6)
Continuation 15050280 · Feb 22, 2016
Continuation 12547406 · Aug 25, 2009
Continuation In Part 12393709 · Feb 26, 2009
Provisional Application 61080184 · Jul 11, 2008
Provisional Application 61031639 · Feb 26, 2008
Related Publication 20190254967A1 · Aug 22, 2019