IP Library › Granted Patent US 11,492,346
Granted Patent B2
US 11,492,346 · App. 16/902,515 · Granted Nov 8, 2022

Benzisoxazole sulfonamide derivatives

Inventors: Ylva Elisabet Bergman Bozikis (Parkville, AU); Michelle Ang Camerino (Parkville, AU); Pei-Pei Kung (San Diego, CA); Paul Anthony Stupple (Melbourne, AU); Scott Channing Sutton (San Diego, CA)
Assignees: Pfizer Inc.; CTXT PTY LTD
C07D413/06A61P35/04A61K45/06C07B2200/13
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Quick Facts
Patent No.
US 11,492,346
App. No.
16/902,515
Granted
Nov 8, 2022
Kind
B2
Abstract

The present invention relates to compounds of formula (I) or pharmaceutically acceptable salts thereof, wherein Ring A, R 1 -R 8 , and n are defined herein. The novel benzisoxazole sulfonamide derivatives are useful in the treatment of abnormal cell growth, such as cancer, in patients. Additional embodiments relate to pharmaceutical compositions containing the compounds and to methods of using the compounds and compositions in the treatment of abnormal cell growth in patients.

Claims (7)

1. A compound

or a pharmaceutically acceptable salt thereof.

2. 2-Methoxy-N-{4-methoxy-6-[(1H-pyrazol-1-yl)methyl]-1,2-benzoxazol-3-yl}benzene-1-sulfonamide.

3. A pharmaceutical composition comprising the compound of claim 1 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier or diluent.

4. A pharmaceutically acceptable salt of 2-methoxy-N-{4-methoxy-6-[(1H-pyrazol-1-yl)methyl]-1,2-benzoxazol-3-yl}benzene-1-sulfonamide.

5. A pharmaceutical composition comprising 2-methoxy-N-{4-methoxy-6-[(1H-pyrazol-1-yl)methyl]-1,2-benzoxazol-3-yl}benzene-1-sulfonamide, and a pharmaceutically acceptable carrier or diluent.

6. A pharmaceutical composition comprising a pharmaceutically acceptable salt of 2-methoxy-N-{4-methoxy-6-[(1H-pyrazol-1-yl)methyl]-1,2-benzoxazol-3-yl}benzene-1- sulfonamide, and a pharmaceutically acceptable carrier or diluent.

Assignments (4)
CHANGE OF ADDRESS Recorded Mar 30, 2023
From: PFIZER INC.
To: PFIZER INC.
Reel/Frame 063192/0915 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 8, 2020
From: MONASH UNIVERSITY
To: CTXT PTY LTD
Reel/Frame 053151/0536 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 8, 2020
From: BRODSKY, OLEG; GREASLEY, SAMANTHA ELIZABETH; HOFFMAN, ROBERT LOUIS; KUMPF, ROBERT ARNOLD; KUNG, PEI-PEI; RICHARDSON, PAUL FRANCIS; SUTTON, SCOTT CHANNING
To: PFIZER INC.
Reel/Frame 053151/0557 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 8, 2020
From: STUPPLE, PAUL ANTHONY; CAMERINO, MICHELLE ANG; BOZIKIS, YLVA ELISABET BERGMAN
To: MONASH UNIVERSITY
Reel/Frame 053154/0246 →
Continuity (4)
Provisional Application 63025278 · May 15, 2020
Provisional Application 62953223 · Dec 24, 2019
Provisional Application 62863199 · Jun 18, 2019
Related Publication 20200399258A1 · Dec 24, 2020
Cited By (3)
US 12,187,732 US 12,365,655 US 12,371,425