IP Library Granted Patent US 11,591,338
Granted Patent B2
US 11,591,338 · App. 17/073,987 · Granted Feb 28, 2023

Pyrrolotriazine compounds as TAM inhibitors

Inventors: Yun-Long Li (Chadds Ford, PA); Xiaozhao Wang (Moorestown, NJ); Chunhong He (Boothwyn, PA)
Assignee: Incyte Corporation
C07D487/04A61K31/53A61P35/00C07D403/04C07D403/14
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Quick Facts
Patent No.
US 11,591,338
App. No.
17/073,987
Granted
Feb 28, 2023
Kind
B2
Abstract

This application relates to compounds of Formula I: or pharmaceutically acceptable salts thereof, which are inhibitors of TAM kinases which are useful for the treatment of disorders such as cancer.

Claims (4)

1. A method for treating a cancer in a patient, said method comprising: administering to the patient a therapeutically effective amount of a compound which is N-(4-(4-Amino-7-(1-isobutyrylpiperidin-4-yl)pyrrolo[1,2-f][1,2,4]triazin-5-yl)phenyl)-1-isopropyl-2,4-dioxo-3-(pyridin-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide, or a pharmaceutically acceptable salt thereof, wherein the cancer is a sarcoma.

2. The method of claim 1 , wherein the sarcoma is selected from rhabdosarcoma, Kaposi sarcoma, and osteosarcoma.

3. The method of claim 1 , wherein the sarcoma is selected from chondrosarcoma, Ewing's sarcoma, osteosarcoma, rhabdomyosarcoma, angiosarcoma, fibrosarcoma, liposarcoma, myxoma, rhabdomyoma, rhabdosarcoma, fibroma, lipoma, harmatoma, and teratoma.

4. The method of claim 1 , wherein the sarcoma is leiomyosarcoma.

Assignments (2)
CORRECTIVE ASSIGNMENT TO CORRECT THE ASSIGNEE'S STATE PREVIOUSLY RECORDED AT REEL: 055470 FRAME: 0517. ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNMENT. Recorded Dec 29, 2021
From: LI, YUN-LONG; WANG, XIAOZHAO; BARBOSA, JOSEPH; BURNS, DAVID M.; FENG, HAO; GLENN, JOSEPH; HE, CHUNHONG; HUANG, TAISHENG; MEI, SONG; ZHUO, JINCONG
To: INCYTE CORPORATION
Reel/Frame 058690/0622 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 10, 2021
From: LI, YUN-LONG; WANG, XIAOZHAO; BARBOSA, JOSEPH; BURNS, DAVID M.; FENG, HAO; GLENN, JOSEPH; HE, CHUNHONG; HUANG, TAISHENG; MEI, SONG; ZHUO, JINCONG
To: INCYTE CORPORATION
Reel/Frame 055470/0517 →
Continuity (7)
Continuation 16559841 · Sep 4, 2019
Continuation 15971017 · May 4, 2018
Continuation 15469975 · Mar 27, 2017
Provisional Application 62438750 · Dec 23, 2016
Provisional Application 62362934 · Jul 15, 2016
Provisional Application 62314066 · Mar 28, 2016
Related Publication 20210147430A1 · May 20, 2021
Cited By (4)
US 12,187,730 US 12,214,036 US 12,318,389 US 12,415,809