IP Library Granted Patent US 12,163,130
Granted Patent B2
US 12,163,130 · App. 17/099,209 · Granted Dec 10, 2024

Compositions and methods for modulating neuronal excitability and motor behavior

Inventors: Anne Schaefer (New York, NY); Paul Greengard (New York, NY); Chan Lek Tan (San Francisco, CA)
Assignees: Icahn School of Medicine at Mount Sinai; The Rockefeller University
C12N15/113A01K67/0275A01K67/0276A61K38/185A61K49/0008G01N33/5058A01K2217/052A01K2217/075A01K2217/203A01K2227/105A01K2267/0356A61P25/00A61P25/08C12N2310/141C12N2310/315C12N2310/321C12N2310/341C12N2310/346C12N2310/3515C12N2310/3521
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Quick Facts
Patent No.
US 12,163,130
App. No.
17/099,209
Granted
Dec 10, 2024
Kind
B2
Abstract

The invention is directed to compositions and methods for treating or reducing the likelihood of the development of epilepsy in an individual. The method comprises administering to the central nervous system of an individual in need of such treatment a therapeutically effective amount of an agent capable of increasing the expression and/or activity of miR-128.

Claims (26)

1. A method for treating or reducing the likelihood of the development of temporal lobe epilepsy in an individual at risk for developing epilepsy, comprising administering to said individual an agent, wherein

said individual has suffered a traumatic brain injury or a brain injury caused by a stroke,

the agent comprises a seed region of microRNA (miR)-128 or a polynucleotide encoding a transcript wherein the transcript comprises the seed region of miR-128, and

the seed region of miR-128 consists of nucleotides 2 through 7 of SEQ ID NO: 1.

2. The method of claim 1 , wherein the agent is administered intrathecally or intranasally.

3. The method of claim 1 , wherein the agent is administered to the central nervous system of the individual.

4. The method of claim 1 , wherein the agent comprises the seed region of miR-128.

5. The method of claim 4 , wherein the agent further comprises a polynucleotide with 90 percent or more sequence identity to SEQ ID NO: 1.

6. The method of claim 4 , wherein the agent further comprises a chemically stabilized polynucleotide.

7. The method of claim 1 , wherein the agent comprises the polynucleotide encoding the transcript.

8. The method of claim 7 , wherein the transcript further comprises a polynucleotide with 90 percent or more sequence identity to SEQ ID NO: 1.

9. The method of claim 7 , wherein the agent further comprises a viral vector.

10. A method for treating or reducing the likelihood of the development of epilepsy in an individual at risk for developing epilepsy, comprising administering to said individual an agent, wherein

said individual has suffered a traumatic brain injury or a brain injury caused by a stroke,

the agent comprises a seed region of microRNA (miR)-128 or a polynucleotide encoding a transcript wherein the transcript comprises the seed region of miR-128, and

the seed region of miR-128 consists of nucleotides 2 through 7 of SEQ ID NO: 1.

11. The method of claim 10 , wherein the agent is administered intrathecally or intranasally.

12. The method of claim 10 , wherein the agent is administered to the central nervous system of the individual.

13. The method of claim 10 , wherein the agent comprises the seed region of miR-128.

14. The method of claim 13 , wherein the agent further comprises a polynucleotide with 90 percent or more sequence identity to SEQ ID NO: 1.

15. The method of claim 13 , wherein the agent further comprises a chemically stabilized polynucleotide.

16. The method of claim 10 , wherein the agent comprises the polynucleotide encoding the transcript.

17. The method of claim 16 , wherein the transcript further comprises a polynucleotide with 90 percent or more sequence identity to SEQ ID NO: 1.

18. The method of claim 16 , wherein the agent further comprises a viral vector.

19. The method of claim 10 , wherein said individual has suffered a traumatic brain injury.

20. The method of claim 10 , wherein said individual has suffered a brain injury caused by a stroke.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 20, 2021
From: TAN, CHAN LEK
To: ROCKEFELLER UNIVERSITY
Reel/Frame 057851/0984 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 27, 2021
From: SCHAEFER, ANNE
To: ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI
Reel/Frame 055051/0765 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 27, 2021
From: GREENGARD, PAUL
To: THE ROCKEFELLER UNIVERSITY
Reel/Frame 055051/0798 →
Continuity (5)
Continuation 16148015 · Oct 1, 2018
Continuation 15032255
Provisional Application 61898952 · Nov 1, 2013
Provisional Application 61896463 · Oct 28, 2013
Related Publication 20210317451A1 · Oct 14, 2021