IP Library Granted Patent US 11,690,907
Granted Patent B2
US 11,690,907 · App. 17/186,941 · Granted Jul 4, 2023

Vaccines formed by virus and antigen conjugation

Inventors: Steven D. Hume (Owensboro, KY); Leigh Burden (Owensboro, KY); Joshua Morton (Evansville, IN); Greg Pogue (Austin, TX); Barry Bratcher (Owensboro, KY); Hugh A. Haydon (Louisville, KY); Carrie A. Simpson (Evansville, IN); Nick Partain (Owensboro, KY); Youngjun Oh (Owensboro, KY); John W. Shepherd (Owensboro, KY); Michael H. Pauly (Del Mar, CA)
Assignee: KBIO HOLDINGS LIMITED
A61K39/215A61K39/145A61K47/6811A61K2039/5256A61K2039/627A61K2039/70
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Quick Facts
Patent No.
US 11,690,907
App. No.
17/186,941
Granted
Jul 4, 2023
Kind
B2
Abstract

Disclosed herein are methods of forming compounds and exemplary stable compounds in the nature of a conjugated compound at refrigerated or room temperature, which in some embodiments comprises an antigen and virus particle mixed in a conjugation reaction to form a conjugate mixture, such that the conditions and steps of forming these products allow for use of the conjugate mixture as a vaccine, including but not limited to use as a vaccine against various pathogens including for treatment of diseases caused by novel coronaviruses (including SARS-COV 2).

Claims (29)

1. A multivalent vaccine, comprising:

a first antigen comprising an influenza hemagglutinin antigen (HA);

a second antigen; and

a carrier comprising a virus particle having surface lysine residues; wherein the first antigen and the second antigen chemically associate with the surface lysine residues.

2. The multivalent vaccine of claim 1 , wherein the second antigen is an influenza HA other than the first antigen.

3. The multivalent vaccine of claim 1 , wherein the vaccine comprises two or more type A hemagglutinin antigens (HAs) and two or more type B HAs.

4. The multivalent vaccine of claim 1 , wherein the second antigen comprises a receptor binding domain of a coronavirus.

5. The multivalent vaccine of claim 4 , wherein the coronavirus is chosen from the group consisting of SARS-CoV-1 and SARS-CoV-2.

6. The multivalent vaccine of claim 5 , wherein the vaccine comprises two or more type A hemagglutinin antigens (HAs) and two or more type B HAs.

7. The multivalent vaccine of claim 1 , wherein the virus particle is a virus.

8. The multivalent vaccine of claim 7 , wherein the virus is a tobacco mosaic virus.

9. The multivalent vaccine of claim 1 , wherein when the vaccine is placed in an unrefrigerated environment at a storage temperature for a time period, an integrity or a concentration of the vaccine at the end of the time period is at least 90% of an initial integrity or an initial concentration of the vaccine, wherein the time period is at least 42 days after a release date of the vaccine.

10. The multivalent vaccine of claim 9 , wherein the storage temperature is at least 20° C.

11. A virus-antigen conjugate, comprising a virus and at least one antigen, wherein the at least one antigen comprises a fusion peptide having a first peptide which comprises a receptor binding domain of a pathogen, and a second peptide wherein the fusion peptide is chemically linked with the virus, and wherein the second peptide is a fragment crystallizable (Fc) region of an antibody capable of binding to a Fc receptor.

12. The conjugate of claim 11 , wherein the conjugate is multivalent, and further comprises at least one influenza hemagglutinin antigen (HA) chosen from the group consisting of type A HA and type B HA.

13. The conjugate of claim 11 , wherein the Fc region is an Fc domain of an IgG1 antibody.

14. The conjugate of claim 13 , further comprising a hinge portion linking the first peptide and the second peptide, wherein the hinge portion contains an amino acid sequence as set forth in SEQ ID NO: 3.

15. The conjugate of claim 14 , wherein the pathogen is a coronavirus having said receptor binding domain.

16. The conjugate of claim 15 , wherein the first peptide contains an amino acid sequence as set forth in SEQ ID NO: 2.

17. The conjugate of claim 15 , wherein the first peptide contains an amino acid sequence as set forth in SEQ ID NO: 8.

18. The conjugate of claim 11 , wherein the virus is a tobacco mosaic virus.

19. The conjugate of claim 18 , wherein the tobacco mosaic virus comprises a N-terminal lysine residue.

20. An antigen, comprising:

a fusion peptide having a first peptide which comprises a receptor binding domain of a coronavirus, and a second peptide wherein the fusion peptide is capable of being chemically linked with a virus particle,

wherein the second peptide is a fragment crystallizable (Fc) region of an antibody capable of binding to a Fc receptor.

21. The antigen of claim 20 , wherein when the antigen is placed in an unrefrigerated environment at a storage temperature for a time period, an integrity or a concentration of the antigen at the end of the time period is at least 90% of an initial integrity or an initial concentration of the antigen, wherein the time period is at least 42 days after a release date of the conjugate.

22. The antigen of claim 21 , wherein the storage temperature is at least 20° C.

23. The antigen of claim 22 , wherein the first peptide contains an amino acid sequence as set forth in SEQ ID NO: 2.

24. The antigen of claim 22 , wherein the first peptide contains an amino acid sequence as set forth in SEQ ID NO: 8.

Assignments (5)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 4, 2026
From: KBIO HOLDINGS LIMITED
To: RP3 INC.
Reel/Frame 075523/0190 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 13, 2021
From: KENTUCKY BIOPROCESSING, INC.
To: KBIO HOLDINGS LIMITED
Reel/Frame 058372/0339 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 4, 2021
From: HUME, STEVEN D.; BURDEN, LEIGH; MORTON, JOSHUA; POGUE, GREG; BRATCHER, BARRY; HAYDON, HUGH A.; SIMPSON, CARRIE A.; PARTAIN, NICK; OH, YOUNGJUN; SHEPHERD, JOHN W.
To: KENTUCKY BIOPROCESSING, INC.
Reel/Frame 056123/0891 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 21, 2021
From: PAULY, MICHAEL H.
To: ZABBIO, INC.
Reel/Frame 055987/0655 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 21, 2021
From: ZABBIO, INC.
To: KENTUCKY BIOPROCESSING, INC.
Reel/Frame 055987/0758 →
Continuity (7)
Continuation In Part 16919943 · Jul 2, 2020
Continuation In Part 16709063 · Dec 10, 2019
Continuation In Part 16437734 · Jun 11, 2019
Provisional Application 63047629 · Jul 2, 2020
Provisional Application 63013284 · Apr 21, 2020
Provisional Application 62683865 · Jun 12, 2018
Related Publication 20210236624A1 · Aug 5, 2021