IP Library Granted Patent US 11,725,004
Granted Patent B2
US 11,725,004 · App. 17/398,155 · Granted Aug 15, 2023

(Cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles

Inventors: Doris Riether (Biberach an der Riss, DE); Florian Paul Christian Binder (Maselheim, DE); Henri Doods (Warthausen, DE); Stephan Georg Mueller (Warthausen, DE); Janet Rachel Nicholson (Oberhoefen, DE); Achim Sauer (Ravensburg-Torkenweiler, DE)
Assignee: Centrexion Therapeutics Corporation
C07D417/12A61K31/422C07D261/04C07D261/14C07D413/02C07D413/12C07D413/14
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Quick Facts
Patent No.
US 11,725,004
App. No.
17/398,155
Granted
Aug 15, 2023
Kind
B2
Abstract

This invention relates to novel (Cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles and their use as CB2 cannabinoid receptor agonists, pharmaceutical compositions containing the same, and their use for the treatment of CB2 receptor mediated disorders or conditions.

Claims (20)

1. A method of treating diabetic neuropathy, comprising administering to a human being an effective amount of a compound selected from the group consisting of

and a pharmaceutically acceptable salt thereof, to treat the diabetic neuropathy.

2. The method of claim 1 , wherein the compound is

3. The method of claim 1 , wherein the compound is administered in the form of a tablet, pill, or capsule.

4. The method of claim 2 , wherein the compound is administered in the form of a tablet, pill, or capsule.

5. A method of treating neuropathic pain due to diabetic peripheral neuropathy, comprising administering to a human being an effective amount of a compound selected from the group consisting of

and a pharmaceutically acceptable salt thereof, to treat the neuropathic pain due to diabetic peripheral neuropathy.

6. The method of claim 5 , wherein the compound is

7. The method of claim 5 , wherein the compound is administered in the form of a tablet, pill, or capsule.

8. The method of claim 6 , wherein the compound is administered in the form of a tablet, pill, or capsule.

9. A method of treating neuropathic pain due to diabetic neuropathy, comprising administering to a human being an effective amount of a compound selected from the group consisting of

and a pharmaceutically acceptable salt thereof, to treat the neuropathic pain due to diabetic neuropathy.

10. The method of claim 9 , wherein the compound is

11. The method of claim 9 , wherein the compound is administered in the form of a tablet, pill, or capsule.

12. The method of claim 10 , wherein the compound is administered in the form of a tablet, pill, or capsule.

13. A method of treating nerve injury-induced neuropathic pain, comprising administering to a human being an effective amount of a compound selected from the group consisting of

and a pharmaceutically acceptable salt thereof, to treat the nerve injury-induced neuropathic pain.

14. The method of claim 13 , wherein the compound is

15. The method of claim 13 , wherein the compound is administered in the form of a tablet, pill, or capsule.

16. The method of claim 14 , wherein the compound is administered in the form of a tablet, pill, or capsule.

Assignments (5)
RELEASE OF SECURITY INTEREST Recorded Nov 21, 2025
From: AVENUE VENTURE OPPORTUNITIES FUND, L.P., AS AGENT
To: CENTREXION THERAPEUTICS CORPORATION
Reel/Frame 073683/0099 →
SECURITY INTEREST Recorded Nov 21, 2025
From: CENTREXION THERAPEUTICS CORPORATION
To: ANKURA TRUST COMPANY, LLC, AS ADMINISTRATIVE AND COLLATERAL AGENT
Reel/Frame 073683/0108 →
SECURITY INTEREST Recorded Jul 12, 2023
From: CENTREXION THERAPEUTICS CORPORATION
To: AVENUE VENTURE OPPORTUNITIES FUND, L.P., AS AGENT
Reel/Frame 064256/0125 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 24, 2023
From: BOEHRINGER INGELHEIM INTERNATIONAL GMBH
To: CENTREXION THERAPEUTICS CORPORATION
Reel/Frame 062792/0719 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 24, 2023
From: RIETHER, DORIS; BINDER, FLORIAN PAUL CHRISTIAN; DOODS, HENRI; MUELLER, STEPHAN GEORG; NICHOLSON, JANET RACHEL; SAUER, ACHIM
To: BOEHRINGER INGELHEIM INTERNATIONAL GMBH
Reel/Frame 062856/0726 →
Priority Claims (1)
EP 13168165 · May 17, 2013 · regional
Continuity (5)
Continuation 16749412 · Jan 22, 2020
Continuation 16143523 · Sep 27, 2018
Continuation 15491035 · Apr 19, 2017
Continuation 14891051
Related Publication 20220135554A1 · May 5, 2022
Cited By (1)
US 12,344,601