IP Library › Granted Patent US 7,745,583
Granted Patent B2
US 7,745,583 · App. 12/612,060 · Granted Jun 29, 2010

Anti-myostatin antibodies

Assignee: Eli Lilly and Company
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Quick Facts
Patent No.
US 7,745,583
App. No.
12/612,060
Granted
Jun 29, 2010
Kind
B2
Abstract

A neutralizing epitope is identified within amino acids 40-64 of the mature form of human myostatin. Antibodies that bind this epitope with high affinity preferentially bind GDF-8 over GDF-11 and may be chimeric, humanized or fully human antibodies, immunoconjugates of the antibodies or antigen-binding fragments thereof. The antibodies of the invention are useful for increasing muscle mass, increasing hone density, or for the treatment of various disorders in mammalian and avian species.

Claims (27)

1. A monoclonal antibody comprising a light chain variable region (LCVR) and a heavy chain variable region (HCVR), wherein said LCVR comprises:

a) a peptide at CDRL1 with SEQ ID NO: 27, 28 or 29

b) a peptide at CDRL2 with SEQ ID NO: 30, and

c) a peptide at CDRL3 with SEQ ID NO: 58,

and wherein said HCVR comprises:

a) a peptide at CDRH1 with SEQ ID NO: 59,

b) a peptide at CDRH2 with SEQ ID NO: 60, and

c) a peptide at CDRH3 with SEQ ID NO: 61.

2. The antibody of claim 1 , wherein the antibody is a full-length antibody, a substantially intact antibody, a Fab fragment, a F(ab′)2 fragment or a single chain Fv fragment.

3. A monoclonal antibody comprising a light chain variable region (LCVR) and a heavy chain variable region (HCVR), wherein said LCVR comprises:

a) a peptide at CDRL1 with SEQ ID NO: 27,

b) a peptide at CDRL2 with SEQ ID NO: 30, and

c) a peptide at CDRL3 with SEQ ID NO: 31,

and wherein said HCVR comprises:

a) a peptide at CDRH1 with SEQ ID NO: 37,

b) a peptide at CDRH2 with SEQ ID NO: 43, and

c) a peptide at CDRH3 with SEQ ID NO: 48.

4. The antibody of claim 3 , wherein the antibody is a full-length antibody, a substantially intact antibody, a Fab fragment, a F(ab′)2 fragment or a single chain Fv fragment.

5. A monoclonal antibody comprising a light chain variable region (LCVR) and a heavy chain variable region (HCVR), wherein said LCVR comprises:

a) a peptide at CDRL1 with SEQ ID NO: 27,

b) a peptide at CDRL2 with SEQ ID NO: 30, and

c) a peptide at CDRL3 with SEQ ID NO: 33,

and wherein said HCVR comprises:

a) a peptide at CDRH1 with SEQ ID NO: 36

b) a peptide at CDRH2 with SEQ ID NO: 45, and

c) a peptide at CDRH3 with SEQ ID NO: 51.

6. The antibody of claim 5 , wherein the antibody is a full-length antibody, a substantially intact antibody, a Fab fragment, a F(ab′)2 fragment or a single chain Fv fragment.

Continuity (5)
Continuation 1206666400
Provisional Application 6072606200 · Oct 12, 2005
Provisional Application 6072523500 · Oct 11, 2005
Provisional Application 6072467000 · Oct 6, 2005
Related Publication 20100087631A1 · Apr 8, 2010