IP Library Granted Patent US 8,008,319
Granted Patent B2
US 8,008,319 · App. 12/353,683 · Granted Aug 30, 2011

Treatment of colorectal polyps with imidazoquinoline derivatives

Assignee: Meda Pharma GmbH & Co. KG
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Quick Facts
Patent No.
US 8,008,319
App. No.
12/353,683
Granted
Aug 30, 2011
Kind
B2
Abstract

The invention relates to treating colorectal polyps and precancercerous colorectal changes by topical administration of immunomodulating drugs of the imidazoquinoline family, such as imiquimod (1-(2-methylpropyl)-1H-imidazo[4,5-c]quinolin-4-amine), resiquimod (4-amino-α,α-dimethyl-2-ethoxymethyl-1H-imidazo[4,5-c]quinoline-1-ethanol), sotirimod (2-methyl-1-(2-methylpropyl)-1H-imidazo[4,5-c][1,5]naphthyridin-4-amine).

Claims (15)

1. A method of treatment of colorectal polyps/polyposis by application of an imidazoquinoline derivative selected from the group consisting of imiquimod, resiquimod and sotirimod.

2. The method of treatment according to claim 1 , wherein the patient is a HIV or immunocompromised patient.

3. The method according to claim 1 , wherein the imidazoquinoline derivative is administered topically, in form of a solution, cream or foam.

4. The method according to claim 1 , wherein the imidazoquinoline derivative is administered 1-7 times per week for several weeks.

5. The method according to claim 4 , wherein the imidazoquinoline derivative is administered 1-5 times per week for several weeks.

6. A method of treatment of precancerous colorectal changes by application of an imidazoquinoline derivative selected from the group consisting of imiquimod, resiquimod and sotirimod.

7. The method according to claim 6 , wherein the imidazoquinoline derivative is administered 1-7 times per week for several weeks.

8. The method according to claim 7 , wherein the imidazoquinoline derivative is administered 1-5 times per week for several weeks.

9. The method of treatment according to claim 6 , wherein the patient is a HIV or immunocompromised patient.

10. The method according to claim 6 , wherein the imidazoquinoline derivative is administered topically, in form of a solution, cream or foam.

11. A method of adjuvant treatment of colorectal polyps/polyposis by application of an imidazoquinoline derivative selected from the group consisting of imiquimod, resiquimod and sotirimod.

12. The method according to claim 11 , wherein the imidazoquinoline derivative is administered 1-7 times per week for several weeks.

13. The method according to claim 12 , wherein the imidazoquinoline derivative is administered 1-5 times per week for several weeks.

14. The method of treatment according to claim 11 , wherein the patient is a HIV or immunocompromised patient.

15. The method according to claim 11 , wherein the imidazoquinoline derivative is administered topically, in form of a solution, cream or foam.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 26, 2009
From: MAUS, JOACHIM; SZELENYI, ISTVAN; PETZOLD, URSULA
To: MEDA PHARMA GMBH & CO. KG
Reel/Frame 022454/0964 →
Continuity (2)
Provisional Application 61006459 · Jan 15, 2008
Related Publication 20090182005A1 · Jul 16, 2009