IP Library Granted Patent US 8,030,331
Granted Patent B2
US 8,030,331 · App. 12/899,542 · Granted Oct 4, 2011

Allosteric modulators of metabotropic glutamate receptors

Assignee: Addex Pharma SA
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Quick Facts
Patent No.
US 8,030,331
App. No.
12/899,542
Granted
Oct 4, 2011
Kind
B2
Abstract

The present invention relates to new compounds of formula (I) wherein A, B, P, Q, W, R 1 and R 2 are defined in the description; invention compounds are useful in the prevention or treatment of central nervous system disorders as well as other disorders modulated by mGluR5 receptors.

Claims (8)

1. A compound selected from the group consisting of:

(4-Fluoro-phenyl)-[(S)-3-(3-pyridin-3-yl-[1,2,4]oxadiazol-5-yl)-piperidin-1-yl]-methanone;

(4-Fluoro-phenyl)-[(S)-3-(3-pyridin-4-yl-[1,2,4]oxadiazol-5-yl)-piperidin-1-yl]-methanone; and

(4-Fluoro-phenyl)-[(S)-3-(3-pyridin-2-yl-[1,2,4]oxadiazol-5-yl)-piperidin-1-yl]-methanone;

or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising a compound of claim 1 and a pharmaceutically acceptable carrier.

3. A method for treating a mammal suffering from Schizophrenia, Delusional Disorder, Schizoaffective Disorder, Schizophreniform Disorder, or Substance-Induced Psychotic Disorder, the method comprising administering a compound of claim 1 to the mammal.

4. The method of claim 3 , wherein the method is a method of treating schizophrenia.

Priority Claims (1)
GB 0325956.1 · Nov 6, 2003 · national
Continuity (2)
Continuation 10578589
Related Publication 20110112143A1 · May 12, 2011