IP Library Granted Patent US 8,569,308
Granted Patent B2
US 8,569,308 · App. 12/885,245 · Granted Oct 29, 2013

Substituted heteroarylamine carboxamide analogs as mGluR5 negative allosteric modulators and methods of making and using the same

Inventors: P. Jeffrey Conn (Brentwood, TN); Craig W. Lindsley (Brentwood, TN); Kyle A. Emmitte (Spring Hill, TN); Charles David Weaver (Franklin, TN); Alice L. Rodriguez (Nashville, TN); Andrew S. Felts (Nashville, TN); Carrie K. Jones (Nashville, TN); Brittney S. Bates (Nashville, TN)
Assignee: Vanderbilt University
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Quick Facts
Patent No.
US 8,569,308
App. No.
12/885,245
Granted
Oct 29, 2013
Kind
B2
Abstract

Disclosed are negative allosteric modulators of the metabotropic glutamate receptor subtype 5 (mGluR5); synthetic methods for making the compounds; pharmaceutical compositions comprising the compounds; and methods of treating neurological and psychiatric disorders associated with glutamate dysfunction using the compounds and compositions. This abstract is intended as a scanning tool for purposes of searching in the particular art and is not intended to be limiting of the present invention.

Claims (4)

1. A compound having the following structure,

or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising a compound having the following structure,

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 13, 2012
From: CONN, P JEFFREY; LINDSLEY, CRAIG W.; EMMITTE, KYLE A.; WEAVER, CHARLES DAVID; RODRIGUEZ, ALICE L.; FELTS, ANDREW S.; JONES, CARRIE K.; BATES, BRITTNEY S.
To: VANDERBILT UNIVERSITY
Reel/Frame 027849/0815 →
CONFIRMATORY LICENSE Recorded Mar 15, 2011
From: VANDERBILT UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 025954/0555 →
Continuity (2)
Provisional Application 61243378 · Sep 17, 2009
Related Publication 20110172247A1 · Jul 14, 2011